Title:
ピロリジン化合物を調製するためのプロセス
Document Type and Number:
Japanese Patent JP7121794
Kind Code:
B2
Abstract:
Processes for preparing 5,5-dimethyl-3-methylenepyrrolidin-2-one, (S)-3,5,5-trimethylpyrrolidine-2-one, (R)-3,5,5-trimethylpyrrolidine-2-one, (S)-2,4,4-trimethylpyrrolidine, and (R)-2,4,4-trimethylpyrrolidine, and their salt forms are disclosed.
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Inventors:
Angel, Paul Tee.
Lewandowski, Berenice
Littler, Benjamin Jay.
Nugent, William A.
Smith, David
Studley, John
Hughes, Robert M.
Lewandowski, Berenice
Littler, Benjamin Jay.
Nugent, William A.
Smith, David
Studley, John
Hughes, Robert M.
Application Number:
JP2020505238A
Publication Date:
August 18, 2022
Filing Date:
August 02, 2018
Export Citation:
Assignee:
VERTEX PHARMACEUTICALS INCORPORATED
International Classes:
C07D207/06; C07D207/267
Domestic Patent References:
JP2017530167A | ||||
JP2019529490A | ||||
JP2020500906A | ||||
JP2013545744A | ||||
JP2013515746A |
Other References:
LAI, John T. et al.,J.Org.Chem.,1980年,45,1513-1514
LIND, Hanns et al.,Tetrahedron Lett.,1980年,21,119-120
LIND, Hanns et al.,Tetrahedron Lett.,1980年,21,119-120
Attorney, Agent or Firm:
Shusaku Yamamoto
Morishita Natsuki
Morishita Natsuki