プロリルヒドロキシラーゼ阻害剤

Title:

プロリルヒドロキシラーゼ阻害剤

Document Type and Number:

Japanese Patent JP2011507894

Kind Code:

A

Abstract:

The invention described herein relates to certain 4-oxo-2-thioxo-1,2,3,4-tetrahydro-7-quinazolinecarboxamide derivatives of formula (I) which are antagonists of HIF prolyl hydroxylases and are useful for treating diseases benefiting from the inhibition of this enzyme, anemia being one example.

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Inventors:

Dimitar Be Gochev
Gian Jin
Wang Young Hui

Application Number:

JP2010539849A

Publication Date:

March 10, 2011

Filing Date:

December 19, 2008

Export Citation:

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Assignee:

GlaxoSmithKline LLC

International Classes:

C07D401/04; A61K31/517; A61K31/5377; A61P7/06; A61P9/00; A61P9/10; A61P43/00; C07D401/06; C07D401/12; C07D401/14; C07D403/04; C07D403/06; C07D409/14; C07D413/06; C07D417/04; C07D417/06

Attorney, Agent or Firm:

Aoyama Aoi
Takuji Yamada
Michiko Matsutani
Nishino Mitsuru
Mizuhara Masahiro

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