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Title:
PDE4インヒビターとしてのピラゾロン誘導体
Document Type and Number:
Japanese Patent JP5529010
Kind Code:
B2
Abstract:
Fixed combination, non-fixed combination or kit of parts comprising 1-(2-{4-[3-(3,4-dimethoxyphenyl)-4,4-dimethyl-5-oxo-4,5-dihydro-1H-pyrazol-1-yl]piperidin-1-yl}-2-oxoethyl)pyrrolidine-2,5-dione, pioglitazone or a pharmaceutically acceptable salt of pioglitazone, and at least one pharmaceutically acceptable auxiliary.

Inventors:
Beate Schmidt
Christian Schoeffler
Jürgen Fortz
Martin Pefeit
Rolf-Peter Hummel
Armin Hazelmann
Christoph Zitt
Andrea Wolsen
Degenhard Marx
Hans-Peter Cry
Deborah Okkerto
Anke Heuser
Johannes A. M. Christians
Hert Jan Sterk
Viromp Pabe Menge
Application Number:
JP2010507909A
Publication Date:
June 25, 2014
Filing Date:
May 14, 2008
Export Citation:
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Assignee:
Takeda GmbH
International Classes:
C07D401/14; A61K31/454; A61K31/5377; A61K31/541; A61K45/00; A61K45/06; A61P11/00; A61P11/02; A61P11/06; A61P43/00; C07D405/14; C07D411/14; C07D413/14
Domestic Patent References:
JP2006169138A
JP2005538140A
JP2007504123A
Foreign References:
WO2005075456A1
Attorney, Agent or Firm:
Toshio Yano
Takuya Kuno
Hiroshi Sugimoto
Takahashi
Kimihiro Hoshi
Hiroyasu Ninomiya
Einzel Felix-Reinhard



 
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