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Title:
QUINOLINE DERIVATIVES FOR USE IN THE TREATMENT OF INFLAMMATORY DISEASES
Document Type and Number:
Japanese Patent JP2023052265
Kind Code:
A
Abstract:
To provide novel quinoline derivatives which are efficient for treating and/or preventing inflammatory diseases, as well as novel therapeutic uses of quinoline derivatives for inflammatory diseases.SOLUTION: The present invention provides a compound of formula (I) for use in treating and/or preventing inflammatory diseases, which is exemplified by 8-chloro-5-(3-(piperidin-1-yl)propoxy)-N-(4-(trifluoromethyl)pyridin-2-yl)quinolin-2-amine, 4-(2-((8-chloro-2-(4-(trifluoromethoxy)phenoxy)quinoline-5-yl)oxy)ethyl)morpholine, or the like.SELECTED DRAWING: None

Inventors:
Jamal Tazi
Romantic Najiman
Florence Moutou
Didier Scheller
Karim Shevri
Michael Hahn
Application Number:
JP2023001382A
Publication Date:
April 11, 2023
Filing Date:
January 06, 2023
Export Citation:
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Assignee:
Avivax
Center National de la Recherche Scientific
Anstitut Curie
Universite de Montpellier
International Classes:
C07D215/38; A61K31/47; A61K31/4709; A61K31/496; A61K31/497; A61K31/5377; A61K31/661; A61K31/675; A61P29/00; C07D215/22; C07D401/04; C07D401/12; C07D401/14; C07F9/60; C12N15/11; C12Q1/6851; C12Q1/686
Attorney, Agent or Firm:
Hiroshi Murakami