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Patent Searching and Data


Title:
Substitution imidazo quinoxaline
Document Type and Number:
Japanese Patent JP6168773
Kind Code:
B2
Abstract:
The present invention relates to substituted imidazoquinoxaline compounds of general formula (I) as inhibitors of Mps-1 Kinase or TTK, and being active against inflammation and cancer.

Inventors:
Marx Copitz
Benjamin badder
Wolf Boehmer
Berthold Cleft
Philip Lienau
Tobias Marquarto
Stephan precht
Gerhard Gee Meister
Christoph Bakescheid-Gerlach
Application Number:
JP2012507628A
Publication Date:
July 26, 2017
Filing Date:
April 24, 2010
Export Citation:
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Assignee:
Bayer Intellectual Property GmbH
International Classes:
C07D487/04; A61K31/4985; A61K31/506; A61K31/5377; A61P35/00; A61P35/02; A61P43/00
Foreign References:
WO2009043934A1
Other References:
European Journal of Medicinal Chemistry,(2009),Vol.44,No.9,pp.3406-3411
Int.J.Immunopathol.Pharmacol.,(2006),Vol.19,No.3,pp.525-538
Bioorg.Med.Chem.,(2004),Vol.12,No.5,pp.1129-1139
Bioorg.Med.Chem.,(2008),Vol.16,No.13,pp.6601-6610
Attorney, Agent or Firm:
Makoto Ono
Kenkyo Kanayama
Mitsuaki Tsubokura
Kazuki Shigemori
Kenji Ando
Hidehiko Ichikawa
Takahiro Aoki
Yoshie Sakurada
Yousuke Kawasaki
Toshikazu Imato
Yoshikazu Iwase
Yasufumi Shiroyama