Title:
Substitution imidazo quinoxaline
Document Type and Number:
Japanese Patent JP6168773
Kind Code:
B2
Abstract:
The present invention relates to substituted imidazoquinoxaline compounds of general formula (I) as inhibitors of Mps-1 Kinase or TTK, and being active against inflammation and cancer.
Inventors:
Marx Copitz
Benjamin badder
Wolf Boehmer
Berthold Cleft
Philip Lienau
Tobias Marquarto
Stephan precht
Gerhard Gee Meister
Christoph Bakescheid-Gerlach
Benjamin badder
Wolf Boehmer
Berthold Cleft
Philip Lienau
Tobias Marquarto
Stephan precht
Gerhard Gee Meister
Christoph Bakescheid-Gerlach
Application Number:
JP2012507628A
Publication Date:
July 26, 2017
Filing Date:
April 24, 2010
Export Citation:
Assignee:
Bayer Intellectual Property GmbH
International Classes:
C07D487/04; A61K31/4985; A61K31/506; A61K31/5377; A61P35/00; A61P35/02; A61P43/00
Foreign References:
WO2009043934A1 |
Other References:
European Journal of Medicinal Chemistry,(2009),Vol.44,No.9,pp.3406-3411
Int.J.Immunopathol.Pharmacol.,(2006),Vol.19,No.3,pp.525-538
Bioorg.Med.Chem.,(2004),Vol.12,No.5,pp.1129-1139
Bioorg.Med.Chem.,(2008),Vol.16,No.13,pp.6601-6610
Int.J.Immunopathol.Pharmacol.,(2006),Vol.19,No.3,pp.525-538
Bioorg.Med.Chem.,(2004),Vol.12,No.5,pp.1129-1139
Bioorg.Med.Chem.,(2008),Vol.16,No.13,pp.6601-6610
Attorney, Agent or Firm:
Makoto Ono
Kenkyo Kanayama
Mitsuaki Tsubokura
Kazuki Shigemori
Kenji Ando
Hidehiko Ichikawa
Takahiro Aoki
Yoshie Sakurada
Yousuke Kawasaki
Toshikazu Imato
Yoshikazu Iwase
Yasufumi Shiroyama
Kenkyo Kanayama
Mitsuaki Tsubokura
Kazuki Shigemori
Kenji Ando
Hidehiko Ichikawa
Takahiro Aoki
Yoshie Sakurada
Yousuke Kawasaki
Toshikazu Imato
Yoshikazu Iwase
Yasufumi Shiroyama