Title:
【発明の名称】5-(3-[エキソビシクロ[2.2.1]ヘプト-2-イルオキシ]-4-メトキシフェニル)-3,4,5,6-テトラヒドロピリミジン-2(1H)-オンの合成の方法および中間体
Document Type and Number:
Japanese Patent JP2960965
Kind Code:
B2
Abstract:
This invention relates to novel processes for preparing the pharmaceutically active compound 5-(3-[(2S)-exo-bicyclo[2.2.1]hept-2-yloxy]-4-methoxyphenyl)-3,4,5,6-tetrahydropyrimidin-2(1H)-one and its corresponding 2R enantiomer and for preparing certain intermediates used in the synthesis of these compounds. It also relates to novel intermediates used in the synthesis of such pharmaceutically active compounds and to other novel compounds that are related to such intermediates.
Inventors:
RAKUURU TOOMASU JII
MAATEIASHOO CHAARUZU DABURYUU
MAATEIASHOO CHAARUZU DABURYUU
Application Number:
JP52423195A
Publication Date:
October 12, 1999
Filing Date:
May 04, 1995
Export Citation:
Assignee:
FUAIZAA INC
International Classes:
C07C69/734; C07C235/34; C07C255/37; C07C259/06; C07C271/16; C07C271/20; C07D239/10; (IPC1-7): C07D239/10
Other References:
【文献】国際公開94/12461(WO,A1)
Attorney, Agent or Firm:
Kazuo Shamoto (4 outside)