Title:
【発明の名称】プロテアーゼ阻害剤
Document Type and Number:
Japanese Patent JP2000500742
Kind Code:
A
Abstract:
Disclosed herein is a compound of the formula known as 2-[N-(N-benzyloxycarbonyl-L-leucinyl)]-2'-[N'-[4-(N,N-dimethylaminomethyl)benzyloxy]carbonyl-L-leucinyl]carbohydrazide; and pharmaceutically acceptable salts, hydrates and solvates thereof.
Inventors:
Car, thomas joseph
Death Jar Race, Rene Louise
Gallagher, Timothy Francis
Halbert, Stacy Marie
Oh, Hija
Scott Kevin, Thompson
Bever, daniel frank
Yamashita, Dennis Shinji
Yen, Jack Wekuo
Death Jar Race, Rene Louise
Gallagher, Timothy Francis
Halbert, Stacy Marie
Oh, Hija
Scott Kevin, Thompson
Bever, daniel frank
Yamashita, Dennis Shinji
Yen, Jack Wekuo
Application Number:
JP51763897A
Publication Date:
January 25, 2000
Filing Date:
October 30, 1996
Export Citation:
Assignee:
SMITHKLINE BEECHAM CORPORATION
International Classes:
A61K31/00; A61K31/16; A61K31/18; A61K31/34; A61K31/343; A61K31/38; A61K31/381; A61K31/41; A61K31/415; A61K31/4155; A61K31/4164; A61K31/4245; A61K31/425; A61K31/426; A61K31/427; A61K31/433; A61K31/44; A61K31/4427; A61K31/443; A61K31/4439; A61K31/445; A61K31/4465; A61K31/4523; A61K31/4525; A61K31/47; A61K31/4709; A61K31/495; A61K31/496; A61K31/4965; A61K31/497; A61K31/535; A61K31/5375; A61K31/5377; A61K31/54; A61K38/00; A61P1/00; A61P1/02; A61P19/00; A61P19/10; A61P29/00; A61P43/00; C07C235/50; C07C243/34; C07C271/22; C07C281/06; C07C311/16; C07C311/29; C07D211/62; C07D213/30; C07D213/71; C07D213/81; C07D215/36; C07D231/18; C07D233/56; C07D241/24; C07D249/10; C07D271/06; C07D271/10; C07D277/20; C07D277/36; C07D277/40; C07D277/56; C07D285/06; C07D285/12; C07D285/125; C07D285/135; C07D295/155; C07D295/20; C07D295/215; C07D307/91; C07D333/34; C07D333/76; C07D401/12; C07D405/12; C07D417/12; C07D417/14; C07K5/062; C07K5/083; C12N9/64; C12Q1/37; G01N33/573; (IPC1-7): C07C235/50; A61P1/02; A61P19/10; A61P29/00; A61P43/00; A61K31/16; A61K31/18; A61K31/343; A61K31/381; A61K31/4245; A61K31/433; A61K31/415; A61K31/4155; A61K31/4164; A61K31/426; A61K31/427; A61K31/44; A61K31/443; A61K31/4439; A61K31/445; A61K31/4525; A61K31/4709; A61K31/497; A61K31/5375; A61K31/5377; A61K31/54; A61K38/00; C07C271/22; C07C281/06; C07C311/29; C07D211/62; C07D213/30; C07D213/71; C07D213/81; C07D215/36; C07D231/18; C07D233/56; C07D249/10; C07D271/06; C07D277/36; C07D277/40; C07D277/56; C07D277/587; C07D285/06; C07D285/135; C07D295/20; C07D307/91; C07D333/34; C07D401/12; C07D405/12; C07D417/12; C07D417/14; C07K5/062; C07K5/083
Attorney, Agent or Firm:
Aoyama Ryo (1 person outside)