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Title:
【発明の名称】チロシン誘導体
Document Type and Number:
Japanese Patent JP2003509488
Kind Code:
A
Abstract:
The compounds of the invention are inhibitors of alpha4 containing integrin-mediated binding to ligands such as VCAM-1 and MAdCAM.

Inventors:
Jackson, David, Wye.
Cyres, Frederick, Sea.
Sutherlin, Daniel, Pea.
Application Number:
JP2001524964A
Publication Date:
March 11, 2003
Filing Date:
September 25, 2000
Export Citation:
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Assignee:
GENENTECH,INC.
International Classes:
A61K31/198; A61K31/27; A61K31/36; A61K31/40; A61K31/402; A61K31/423; A61K31/438; A61K31/44; A61K31/4439; A61K31/4458; A61K31/4462; A61K31/4465; A61K31/45; A61K31/454; A61K31/47; A61K31/472; A61K31/495; A61K31/5375; A61K31/5377; A61P1/00; A61P1/04; A61P1/16; A61P1/18; A61P3/10; A61P5/50; A61P11/00; A61P11/02; A61P11/06; A61P15/14; A61P17/00; A61P17/06; A61P19/02; A61P25/00; A61P29/00; A61P37/02; A61P37/06; A61P43/00; C07C233/87; C07C235/38; C07C237/06; C07C237/20; C07C271/22; C07C271/44; C07C271/46; C07C271/48; C07C271/50; C07C271/54; C07C271/56; C07C271/58; C07C271/66; C07C311/06; C07C311/09; C07C311/53; C07C311/58; C07C323/43; C07C323/59; C07D207/16; C07D207/22; C07D207/28; C07D207/325; C07D211/46; C07D211/60; C07D211/62; C07D211/78; C07D213/75; C07D215/36; C07D217/06; C07D217/14; C07D217/22; C07D231/16; C07D235/06; C07D235/26; C07D241/04; C07D249/18; C07D263/58; C07D277/12; C07D277/20; C07D277/56; C07D295/20; C07D295/205; C07D307/68; C07D317/58; C07D333/20; C07D333/34; C07D333/38; C07D333/40; C07D333/62; C07D333/70; C07D333/72; C07D401/04; C07D417/04; C07D471/10; (IPC1-7): C07C233/87; A61K31/198; A61K31/27; A61K31/36; A61K31/40; A61K31/402; A61K31/423; A61K31/438; A61K31/44; A61K31/4439; A61K31/4458; A61K31/4462; A61K31/4465; A61K31/45; A61K31/454; A61K31/47; A61K31/472; A61K31/495; A61K31/5375; A61K31/5377; A61P1/00; A61P1/04; A61P1/16; A61P1/18; A61P3/10; A61P5/50; A61P11/00; A61P11/02; A61P11/06; A61P15/14; A61P17/00; A61P17/06; A61P19/02; A61P25/00; A61P29/00; A61P37/02; A61P37/06; A61P43/00; C07C235/38; C07C237/06; C07C237/20; C07C271/22; C07C271/44; C07C271/46; C07C271/48; C07C271/50; C07C271/54; C07C271/56; C07C271/58; C07C271/66; C07C311/06; C07C311/09; C07C311/53; C07C323/43; C07C323/59; C07D207/16; C07D207/22; C07D207/325; C07D211/46; C07D211/60; C07D211/62; C07D211/78; C07D213/75; C07D215/36; C07D217/06; C07D231/16; C07D235/06; C07D241/04; C07D249/18; C07D263/58; C07D277/56; C07D295/20; C07D307/68; C07D317/58; C07D333/20; C07D333/38; C07D333/40; C07D333/70; C07D333/72; C07D401/04; C07D417/04; C07D471/10
Domestic Patent References:
JP2001089368A2001-04-03
JP2002509131A2002-03-26
Foreign References:
WO1999036393A11999-07-22
Attorney, Agent or Firm:
Yoshitaka Sonoda (1 outside)