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Title:
トレプロスチニル誘導体ならびにその組成物および使用
Document Type and Number:
Japanese Patent JP7013245
Kind Code:
B2
Abstract:
The present disclosure provides treprostinil derivatives that can act as prodrugs of treprostinil. The treprostinil derivatives can be used to treat any conditions responsive to treatment with treprostinil, including pulmonary hypertension, such as pulmonary arterial hypertension.

Inventors:
Chang Xiao Min
Venkatraman Minakshi S.
Becker Cyrus Kay.
Application Number:
JP2017564668A
Publication Date:
January 31, 2022
Filing Date:
June 14, 2016
Export Citation:
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Assignee:
Corsair Pharma Incorporated
International Classes:
C07C69/675; A61K9/70; A61K31/215; A61K31/337; A61K31/341; A61K31/351; A61P9/00; A61P9/04; A61P9/10; A61P9/12; A61P11/00; A61P11/06; A61P13/12; A61P25/04; A61P35/00; A61P37/04; C07C69/28; C07C69/708; C07C69/712; C07C69/74; C07C69/743; C07C69/75; C07C69/96; C07D305/08; C07D307/24; C07D309/08
Domestic Patent References:
JP2003523935A
JP2014527050A
JP2007501281A
JP2003535132A
Foreign References:
WO2014110491A1
WO2003049676A2
Attorney, Agent or Firm:
Shimizu Hatsushi
Masao Haruna
Hirotaka Yamaguchi
Shun Jinbe
Ryuichi Inoue
Toshimitsu Sato
Koichi Niimi
Tomohiko Kobayashi
Hideki Kodera
Masato Ozeki
Kazuya Kawamoto