Title:
VITALLY INFLUENCING SOFT TERTIARY AMINE ESTER OF CARBOXYLIC ACID
Document Type and Number:
Japanese Patent JPS57106647
Kind Code:
A
Abstract:
Derivatives of known bio-affecting carboxylic acids, their non-toxic pharmaceuticaily acceptable acid addition salts and N-oxides as well as processes for preparing those novel derivatives are disclosed. Those derivatives having the structural formula
wherein R-COO- is the acyloxy residue of a bio-affecting monocarboxylic acid;
Y and Y min are each hydrogen or alkyl; n is zero or one;
R1 and R2 are each inter alia alkyl, alkenyl, aryl, cycloalkyl, cycloalkenyl, aralkyl or alkaryl; and R3 is inter alia hydrogen; or the structural formula
wherein -OOC-R min -COO- is the di(acyloxy) residue of a bio-affecting dicarboxylic acid.
Inventors:
KENESU BII SUROON
Application Number:
JP17373881A
Publication Date:
July 02, 1982
Filing Date:
October 31, 1981
Export Citation:
Assignee:
MERCK & CO INC
International Classes:
A61K31/19; A61K31/215; A61K31/40; A61K31/403; A61K31/404; A61K31/415; A61K31/43; A61K31/44; A61K31/4402; A61K31/4409; A61K31/4418; A61K31/545; A61K31/57; A61P9/12; A61P25/04; A61P29/00; A61P31/04; A61P35/00; C07C67/00; C07C219/00; C07C219/10; C07C219/14; C07C219/28; C07C223/02; C07C227/00; C07C227/08; C07C227/16; C07C227/18; C07C229/00; C07C237/20; C07C291/02; C07C291/04; C07C313/00; C07C323/24; C07C401/00; C07C405/00; C07D207/16; C07D207/20; C07D209/18; C07D209/28; C07D213/80; C07D231/12; C07D231/56; C07D233/60; C07D403/12; C07D473/08; C07D475/04; C07D499/00; C07D499/32; C07D499/44; C07D499/46; C07D499/60; C07D499/62; C07D499/68; C07D499/72; C07D499/74; C07D499/76; C07D499/80; C07D501/20; C07D521/00; C07J7/00; C07J41/00; C07J43/00; (IPC1-7): C07C93/16; C07C93/26; C07C95/08; C07C101/02; C07C103/52; C07C103/76; C07C135/00; C07C149/247; C07C177/00; C07D233/60; C07D403/12; C07D473/08; C07D475/04