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Title:
TLR7/8アンタゴニストおよびそれらの使用
Document Type and Number:
Japanese Patent JP7239554
Kind Code:
B2
Abstract:
The present invention relates to compounds of Formula I and pharmaceutically acceptable compositions thereof, useful as TLR7/8 antagonists.

Inventors:
Scherer, Brian A.
Bulgur, nadia
Orchid
Chen, Shea Oleen
Application Number:
JP2020502368A
Publication Date:
March 14, 2023
Filing Date:
July 17, 2018
Export Citation:
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Assignee:
Merck Patent Gesellschaft mit beschraenkter Haftung
International Classes:
C07D401/04; A61K31/454; A61K31/4545; A61K31/4709; A61K31/498; A61K31/4985; A61K31/5377; A61P1/04; A61P3/10; A61P9/10; A61P13/12; A61P17/06; A61P19/00; A61P19/02; A61P19/06; A61P19/10; A61P25/00; A61P25/16; A61P25/28; A61P29/00; A61P31/04; A61P35/00; A61P37/02; A61P43/00; C07D401/14; C07D403/04; C07D403/14; C07D471/04
Domestic Patent References:
JP1156960A
JP2016539079A
JP2014518892A
JP2014516059A
JP2011529932A
JP2007538085A
JP2008545651A
JP2013534208A
Foreign References:
WO2017106607A1
WO2008031566A2
WO2007114763A1
WO2002030930A2
Attorney, Agent or Firm:
Aoki Atsushi
Shinji Mihashi
Youichi Watanabe
Nakajima Masaru
Tatsunori Ikeda