Title:
An imidazoline derivative, its manufacturing process, and the application to those medicines
Document Type and Number:
Japanese Patent JP6262733
Kind Code:
B2
Abstract:
New imidazoline derivatives represented by formula (I), preparation methods thereof, pharmaceutical compositions comprising such derivatives, and applications of such derivatives in preparing androgen receptor antagonists and medicaments for treating diseases such as prostate cancer.
Inventors:
Lou, Haejun
Sun, Piao Yang
Faye, Hongbo
Gian, Hongjien
One, Haway
Don, Chin
Sun, Piao Yang
Faye, Hongbo
Gian, Hongjien
One, Haway
Don, Chin
Application Number:
JP2015528857A
Publication Date:
January 17, 2018
Filing Date:
August 26, 2013
Export Citation:
Assignee:
SHANGHAI HENGRUI PHARMACEUTICAL CO., LTD.
JIANGSU HENGRUI MEDICINE CO.,LTD.
JIANGSU HENGRUI MEDICINE CO.,LTD.
International Classes:
A61K31/4178; C07D233/86; A61K31/4439; A61K31/454; A61P1/14; A61P13/08; A61P15/10; A61P17/10; A61P17/14; A61P33/08; A61P35/00; A61P43/00; C07D401/04; C07D401/12; C07D403/12; C07D405/12; C07D405/14; C07D409/12
Domestic Patent References:
JP2011068653A |
Foreign References:
CN101817787A | ||||
WO2010118354A1 |
Attorney, Agent or Firm:
Xie Takamine
Tadayuki Motoyama
Tadayuki Motoyama
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