Title:
A new immunomodulator and an anti-inflammatory compound
Document Type and Number:
Japanese Patent JP6207393
Kind Code:
B2
Abstract:
The present invention provides dihydroorotate dehydrogenase inhibitors, methods of preparing them, pharmaceutical compositions containing them and methods of treatment, prevention and/or amelioration of diseases or disorders wherein the inhibition of Dihydroorotate dehydrogenase is known to show beneficial effect.
Inventors:
Musupala Niappan, Mayappan
Bavar, Prasnanto, Casinas
Viswanada, Suricant
Vakaranka, Swarup, Kumar, Vie. Es.
Merica Pudy, Gayatri, Swallow
Bavar, Prasnanto, Casinas
Viswanada, Suricant
Vakaranka, Swarup, Kumar, Vie. Es.
Merica Pudy, Gayatri, Swallow
Application Number:
JP2013508570A
Publication Date:
October 04, 2017
Filing Date:
May 06, 2011
Export Citation:
Assignee:
Incozen Therapeutics Private Limited
Rezen Pharmaceuticals S.A.
Rezen Pharmaceuticals S.A.
International Classes:
C07C235/42; A61K31/167; A61K31/185; A61K31/192; A61K31/343; A61K31/357; A61K31/36; A61K31/404; A61K31/4184; A61K31/44; A61K31/4965; A61K45/00; A61P1/00; A61P1/04; A61P1/16; A61P7/00; A61P11/02; A61P13/12; A61P17/00; A61P17/02; A61P17/06; A61P19/02; A61P19/10; A61P21/02; A61P25/00; A61P25/04; A61P27/02; A61P29/02; A61P31/04; A61P35/00; A61P37/00; A61P37/02; A61P37/06; A61P37/08; A61P43/00; C07C235/84; C07C309/61; C07C317/38; C07C321/28; C07D209/08; C07D213/81; C07D231/56; C07D241/24; C07D307/79; C07D317/58; C07D319/18
Domestic Patent References:
JP5533104A | ||||
JP63295539A | ||||
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POLYMER SCIENCE U.S.S.R.,(1976),V18,N8,pp.2133-2141
ARZNEIMITTELFORSCHUNG DRUG RESEARCH,(1973),V23,N12,pp.1745-1758
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CAplus(STN)[online],レコード番号1953:25381
CAplus(STN)[online],レコード番号1943:542
POLYMER SCIENCE U.S.S.R.,(1976),V18,N8,pp.2133-2141
ARZNEIMITTELFORSCHUNG DRUG RESEARCH,(1973),V23,N12,pp.1745-1758
JOURNAL OF MEDICINAL CHEMISTRY,(1992),V35,N12,pp.2210-2214
JOURNAL OF ORGANIC CHEMISTRY,(1993),58(21),pp.5607-5614
日本化学会誌,(1974),11,pp.2181-2185
PHARMACEUTICAL CHEMISTRY JOURNAL,(2005),39(8),pp.409-412
CURRENT ALZHEIMER RESEARCH,(2007),4(3),pp.315-323
REGISTRY(STN)[online],2006年5月1日,[検索日2016.04.08],CAS登録番号122818-00-2,136071-17-5,882322-26-1
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,(1950),72,pp.153-155
CAplus(STN)[online],レコード番号1953:25381
CAplus(STN)[online],レコード番号1943:542
Attorney, Agent or Firm:
Tatsuya Saito