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Title:
ケモカイン受容体CCR5のモジュレーターとしての新規なピペリジン誘導体
Document Type and Number:
Japanese Patent JP2006514107
Kind Code:
A
Abstract:
Compounds of formula (I) wherein R1, R2R3, R4, Lambda, X, m and n are as defined; compositions comprising them, processes for preparing them and their use in medical therapy them and their use in medical therapy (for example mod ulating CCR 5 receptor activity in a warm blooded animal).

Inventors:
John Cumming
Alan Fall
Colin Fielding
John Oldfield
Howard Tucker
Application Number:
JP2005502630A
Publication Date:
April 27, 2006
Filing Date:
December 18, 2003
Export Citation:
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Assignee:
ASTRAZENECA AKTIEBOLAG
International Classes:
C07D211/24; A61K31/4468; A61K31/4523; A61K31/4545; A61K31/497; A61P1/00; A61P11/00; A61P17/00; A61P17/06; A61P19/00; A61P29/00; A61P31/12; A61P31/18; A61P35/00; A61P37/06; C07D211/58; C07D211/96; C07D401/06; C07D401/12; C07D401/14; C07D405/06; C07D405/12; C07D417/14
Domestic Patent References:
JPH06500093A1994-01-06
JPH11147872A1999-06-02
Foreign References:
WO2001087839A12001-11-22
WO2000076514A12000-12-21
Attorney, Agent or Firm:
Aoyama Aoi
Mitsutaka Iwasaki
Shoji Nakajima