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Title:
ORAL SOLID PREPARATION
Document Type and Number:
Japanese Patent JP2022170891
Kind Code:
A
Abstract:
To provide an oral solid preparation having improved bitterness of a compound A, particularly an orally disintegrating tablet.SOLUTION: An oral solid preparation contains 8-[(3R)-3-aminopiperidine-1-yl]-7-(buta-2-yne-1-yl)-3-methyl-1-[(4-methylquinazoline-2-yl)methyl]-3,7-dihydro-1H-purine-2,6-dione or a pharmaceutically acceptable salt thereof and an anionic polymer.SELECTED DRAWING: None

Inventors:
OKABE KOTA
YAKUWA TAKUSHI
Application Number:
JP2021077170A
Publication Date:
November 11, 2022
Filing Date:
April 30, 2021
Export Citation:
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Assignee:
NISSHIN SEIYAKU KK
International Classes:
A61K31/522; A61K9/20; A61K47/18; A61K47/26; A61K47/32; A61K47/36; A61K47/38; A61K47/42
Attorney, Agent or Firm:
Hisato Ohgushi
Mariko Tsuji
Toshihiko Sato