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Title:
フルクトースおよび関連する炭水化物ならびにポリオールを有するp-ボロノフェニルアラニン錯体
Document Type and Number:
Japanese Patent JP4643017
Kind Code:
B2
Abstract:
The present invention is directed to salt-free and essentially salt-free p-boronophenylalanine-carbohydrate or p-boronophenylalanine-polyol complexes, as well as methods for making such compounds. In addition, the present invention provides methods for substantially solubilizing freeze-dried p-boronophenylalanine-carbohydrate and p-boronophenylalanine-polyol complexes. The present invention further provides compositions and methods for enhancing the solubility of boronophenylalanine.

Inventors:
Sur, Brian
Spiel Vogel, David
Head, gerald
Application Number:
JP2000607637A
Publication Date:
March 02, 2011
Filing Date:
March 24, 2000
Export Citation:
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Assignee:
Glicocin Pharmaceuticals, Inc.
International Classes:
C07F5/02; C07B59/00; C07H23/00; C07H1/00
Domestic Patent References:
JP11255773A
Foreign References:
US5492900
Attorney, Agent or Firm:
Yusuke Hiraki
Satoshi Fujita
Ishii Teiji