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Title:
The pyrazolo Naphthyridinones derivative as METAP2 inhibitor (2 type methionine amino peptidase)
Document Type and Number:
Japanese Patent JP2016515541
Kind Code:
A
Abstract:
本発明は、式(I)のピラゾロナフチリジノン誘導体、それらの調製およびそれらの2型メチオニンアミノペプチターゼ(hMETAP2)選択的阻害剤としての治療的使用に関する。【化1】

Inventors:
Natalie Guillo
Valerie Martin
Application Number:
JP2016503675A
Publication Date:
May 30, 2016
Filing Date:
March 21, 2014
Export Citation:
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Assignee:
SANOFI
International Classes:
C07D471/14; A61K31/4375; A61K31/444; A61K31/4709; A61K31/496; A61K31/506; A61K31/5377; A61K31/551; A61P1/16; A61P3/04; A61P11/00; A61P15/00; A61P17/06; A61P19/00; A61P19/02; A61P27/02; A61P29/00; A61P33/02; A61P35/00; A61P37/02; A61P43/00
Foreign References:
WO2007032466A12007-03-22
WO2012154678A12012-11-15
Attorney, Agent or Firm:
Junji Yuda
Noriyuki Takebayashi