Title:
4,4-DIFLUORO-1,2,3,4-TETRAHYDRO-5H-1-BENZAZEPINE DERIVATIVE OR SALT THEREOF
Document Type and Number:
WIPO Patent Application WO/2004/096775
Kind Code:
A1
Abstract:
A novel 4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepine derivative represented by the following formula (I) or a pharmaceutically acceptable salt of the derivative. They are useful as a therapeutic or preventive agent for night pollakisuria and/or diabetes insipidus.
Inventors:
KOSHIO HIROYUKI (JP)
TSUKAMOTO ISSEI (JP)
KAKEFUDA AKIO (JP)
AKAMATSU SEIJIRO (JP)
SAITOH CHIKASHI (JP)
TSUKAMOTO ISSEI (JP)
KAKEFUDA AKIO (JP)
AKAMATSU SEIJIRO (JP)
SAITOH CHIKASHI (JP)
Application Number:
PCT/JP2004/005998
Publication Date:
November 11, 2004
Filing Date:
April 26, 2004
Export Citation:
Assignee:
YAMANOUCHI PHARMA CO LTD (JP)
KOSHIO HIROYUKI (JP)
TSUKAMOTO ISSEI (JP)
KAKEFUDA AKIO (JP)
AKAMATSU SEIJIRO (JP)
SAITOH CHIKASHI (JP)
KOSHIO HIROYUKI (JP)
TSUKAMOTO ISSEI (JP)
KAKEFUDA AKIO (JP)
AKAMATSU SEIJIRO (JP)
SAITOH CHIKASHI (JP)
International Classes:
A61P13/02; A61P43/00; C07D223/16; (IPC1-7): C07D223/16; C07D401/06; C07D401/12; C07D403/06; C07D403/12; C07D417/06; A61K31/55; A61P13/02; A61P43/00
Domestic Patent References:
WO1995006035A1 | 1995-03-02 | |||
WO1998039325A1 | 1998-09-11 |
Foreign References:
JPH09221476A | 1997-08-26 | |||
JPH08301848A | 1996-11-19 |
Other References:
See also references of EP 1619185A4
None
None
Attorney, Agent or Firm:
Nagai, Shozo c/o Astellas Pharma Inc. (Intellectual Property 3-11, Nihonbashi-Honcho 2-chom, Chuo-ku Tokyo, JP)
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