Title:
A2B ADENOSINE RECEPTOR ANTAGONISTS
Document Type and Number:
WIPO Patent Application WO2003042214
Kind Code:
A3
Abstract:
Disclosed are novel compounds of the Formula I or Formula II that are A2B adenosine receptor antagonists, useful for treating various disease states, including asthma and diarrhea.
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Inventors:
KALLA RAO
PERRY THAO
ELZEIN ELFATIH
VARKHEDKAR VAIBHAV
LI XIAOFEN
IBRAHIM PRABHA
PALLE VENKATA
XIAO DENGMING
ZABLOCKI JEFF
PERRY THAO
ELZEIN ELFATIH
VARKHEDKAR VAIBHAV
LI XIAOFEN
IBRAHIM PRABHA
PALLE VENKATA
XIAO DENGMING
ZABLOCKI JEFF
Application Number:
PCT/US2002/035880
Publication Date:
March 04, 2004
Filing Date:
November 08, 2002
Export Citation:
Assignee:
CV THERAPEUTICS INC (US)
International Classes:
A61K31/522; A61K31/53; A61P1/12; A61P3/10; A61P9/00; A61P9/10; A61P11/06; A61P25/16; A61P25/28; C07D473/04; A61P27/02; A61P35/00; A61P43/00; C07D285/08; C07D473/00; C07D473/06; C07D473/08; (IPC1-7): C07D473/00; C07D473/06; C07D473/08; A61K31/52; A61P1/12; A61P11/06; A61P25/16; A61P25/28; A61P35/00
Domestic Patent References:
| WO1995011681A1 | 1995-05-04 | |||
| WO2000073307A2 | 2000-12-07 |
Foreign References:
| US4879296A | 1989-11-07 | |||
| EP1084710A1 | 2001-03-21 | |||
| US5532368A | 1996-07-02 |
Other References:
JACOBSON K A ET AL: "1,3-DIALKYLXANTHINE DERIVATIVES HAVING HIGH POTENCY AS ANTAGONISTS AT HUMAN A2B ADENOSINE RECEPTORS", DRUG DEVELOPMENT RESEARCH, NEW YORK, NY, US, vol. 47, no. 1, 1999, pages 45 - 53, XP000942540, ISSN: 0272-4391
KUZ'MENKO I I ET AL: "REACTIONS OF THEOPHYLLINES. CHEMICAL CONVERSIONS OF 8-AMINOTHEOPHYLLINATES", CHEMISTRY OF HETEROCYCLIC COMPOUNDS (A TRANSLATION OF KHIMIYA GETEROTSIKLICHESKIKH SOEDINENII), PLENUM PRESS CO., NEW YORK, NY, US, vol. 36, no. 8, 2000, pages 963 - 970, XP001146936, ISSN: 0009-3122
KUZ'MENKO I I ET AL: "REACTIONS OF THEOPHYLLINES. CHEMICAL CONVERSIONS OF 8-AMINOTHEOPHYLLINATES", CHEMISTRY OF HETEROCYCLIC COMPOUNDS (A TRANSLATION OF KHIMIYA GETEROTSIKLICHESKIKH SOEDINENII), PLENUM PRESS CO., NEW YORK, NY, US, vol. 36, no. 8, 2000, pages 963 - 970, XP001146936, ISSN: 0009-3122
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