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Patent Searching and Data


Title:
ADENOSINE DERIVATIVE
Document Type and Number:
WIPO Patent Application WO/1999/048903
Kind Code:
A1
Abstract:
An adenosine derivative acting selectively on P3-like receptor (purine receptor 3-like substance). Because of being capable of binding selectively to P3-like receptor, this adenosine derivative is usable in screening P3-like receptor and substances having the action thereof and, in its turn, useful in studying pharmacological, biochemical and physiological effects and mechanisms of purine receptors.

Inventors:
MATSUDA AKIRA (JP)
NAKATA HIROYASU (JP)
SAITOH YOSHIKO (JP)
Application Number:
PCT/JP1999/001459
Publication Date:
September 30, 1999
Filing Date:
March 23, 1999
Export Citation:
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Assignee:
MATSUDA AKIRA (JP)
NAKATA HIROYASU (JP)
SAITOH YOSHIKO (JP)
International Classes:
C07H19/16; G01N33/566; (IPC1-7): C07H19/16; G01N33/15
Other References:
MATSUDA A., ET AL.: "NUCLEOSIDES AND NUCLEOTIDES. 177. 9-(6,7-DIDEOXY-BETA-D-ALLO-HEPT-5-YNOFURANOSYL)ADENINE: A SELECTIVE AND POTENT LIGAND FOR P3 PURINOCEPTOR-LIKE PROTEIN.", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, US, vol. 41., no. 15., 16 July 1998 (1998-07-16), US, pages 2676 - 2678., XP002920989, ISSN: 0022-2623, DOI: 10.1021/jm9802822
SHINOZUKA K., BJUR R. A., WESTFALL D. P.: "CHARACTERIZATION OF PREJUNCTIONAL PURINOCEPTORS ON ADRENERGIC NERVES OF THE RAT CAUDAL ARTERY.", NAUNYN-SCHMIEDEBERG'S ARCHIVES OF PHARMACOLOGY, SPRINGER, DE, vol. 338., 1 January 1988 (1988-01-01), DE, pages 221 - 227., XP002920990, ISSN: 0028-1298, DOI: 10.1007/BF00173391
Attorney, Agent or Firm:
Hirose, Takayoshi (Nishitenma 5-chome Kita-ku, Osaka-shi Osaka, JP)
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