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Title:
AMINE COMPOUND FOR INHIBITING SSAO/VAP-1 AND USE THEREOF IN MEDICINE
Document Type and Number:
WIPO Patent Application WO/2019/024924
Kind Code:
A1
Abstract:
The present invention relates to an amine compound for inhibiting semicarbazide-sensitive amine oxidase (SSAO) and/or vascular adhesion protein-1 (VAP-1) inhibitors and use thereof in medicine, and further relates to a pharmaceutical composition comprising the amine compound. Said compound and pharmaceutical composition can be used for treating inflammation and/or inflammation related diseases, diabetes and/or diabetes related diseases, psychiatric disorders, ischemic diseases, vascular diseases, fibrosis or tissue transplant rejection.

Inventors:
GU ZHENG (CN)
LI JIANHAO (CN)
LI ZHENG (CN)
WANG WEIHUA (CN)
QIN HAOXIONG (CN)
CUI YUNZENG (CN)
WANG XULI (CN)
YU SHUNA (CN)
ZHANG YINGJUN (CN)
Application Number:
PCT/CN2018/098563
Publication Date:
February 07, 2019
Filing Date:
August 03, 2018
Export Citation:
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Assignee:
SUNSHINE LAKE PHARMA CO LTD (CN)
International Classes:
A61K31/135; C07C211/29; A61P29/00; C07C211/26; C07C217/54
Foreign References:
CN108341752A2018-07-31
US20070293548A12007-12-20
CN104520268A2015-04-15
CN1921841A2007-02-28
CN101917845A2010-12-15
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