AMINOHETEROARYL COMPOUNDS AS PROTEIN KINASE INHIBITORS

WIPO Patent Application WO2004076412

A3

Aminopyridine and aminopyrazine compounds of formula (1), compositions including these compounds, and methods of their use are provided. Preferred compounds of formula 1 have activity as protein kinase inhibitors, including as inhibitors of c-MET.

CUI JINGJONG JEAN (US)
BHUMRALKAR DILIP (US)
BOTROUS IRINY (US)
CHU JI YU (US)
FUNK LEE A (US)
HANAU CATHLEEN ELIZABETH (US)
HARRIS JR G DAVIS (US)
JIA LEI (US)
JOHNSON JOANNE (US)
KOLODZIEJ STEPHEN A (US)
KUNG PEI-PEI (US)
LI XIAOYUAN SHARON (US)
LIN JASON QISHEN (US)
MENG JERRY JIALUN (US)
NAMBU MITCHELL DAVID (US)
NELSON CHRISTOPHER G (US)
PAIRISH MASON ALAN (US)
SHEN HONG (US)
TRAN-DUBE MICHELLE (US)
WALTER ALLISON (US)
ZHANG FANG-JIE (US)
ZHANG ZENNIFER (US)

PCT/US2004/005495

December 29, 2004

February 26, 2004

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SUGEN INC (US)
CUI JINGJONG JEAN (US)
BHUMRALKAR DILIP (US)
BOTROUS IRINY (US)
CHU JI YU (US)
FUNK LEE A (US)
HANAU CATHLEEN ELIZABETH (US)
HARRIS JR G DAVIS (US)
JIA LEI (US)
JOHNSON JOANNE (US)
KOLODZIEJ STEPHEN A (US)
KUNG PEI-PEI (US)
LI XIAOYUAN SHARON (US)
LIN JASON QISHEN (US)
MENG JERRY JIALUN (US)
NAMBU MITCHELL DAVID (US)
NELSON CHRISTOPHER G (US)
PAIRISH MASON ALAN (US)
SHEN HONG (US)
TRAN-DUBE MICHELLE (US)
WALTER ALLISON (US)
ZHANG FANG-JIE (US)
ZHANG ZENNIFER (US)

A61K31/44; A61K31/496; A61K31/4965; A61K31/497; C07D211/72; C07D213/73; C07D401/00; C07D401/12; C07D403/00; C07D405/00; C07D409/00; C07D411/00; C07D413/00; C07D413/12; C07D417/00; C07D419/00; A61K; C07D; (IPC1-7): A61K31/4965; C07D401/00; C07D403/00; C07D405/00; C07D409/00; C07D411/00; C07D413/00; C07D417/00; C07D419/00; C07D211/72

WO2003000666A1

2003-01-03

See also references of EP 1603570A4

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