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Title:
ANTI-HBV AGENT
Document Type and Number:
WIPO Patent Application WO/2020/255425
Kind Code:
A1
Abstract:
This anti-HBV agent contains a compound represented by general formula (I) or a compound represented by general formula (II), or a salt thereof.

Inventors:
KOJIMA SOICHI (JP)
FURUTANI YUTAKA (JP)
DOHMAE NAOSHI (JP)
OGAWA KENJI (JP)
ICHIKAWA YASUE (JP)
NIWA TAKASHI (JP)
WATANABE KENJI (JP)
HOSOYA TAKAMITSU (JP)
KANAYAMA YOSUKE (JP)
WATANABE YASUYOSHI (JP)
HIRANO YOSHINORI (JP)
SHIROUZU MIKAKO (JP)
IWASAKI WAKANA (JP)
Application Number:
PCT/JP2019/024847
Publication Date:
December 24, 2020
Filing Date:
June 21, 2019
Export Citation:
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Assignee:
RIKEN (JP)
International Classes:
A61K31/167; A61K31/4409; A61K31/4468; A61K31/505; A61P31/20; C07C235/84; C07C247/16; C07C247/18; C07C255/60; C07C323/42; C07D211/58; C07D213/74; C07D239/42; C07F5/04; C07F7/12; G01N33/15; G01N33/50
Domestic Patent References:
WO2004022585A12004-03-18
Foreign References:
JP2002521437A2002-07-16
JP2019112326A2019-07-11
Other References:
LI CHUANG, REN SHI-FANG, HOU JUN-LI, YI HUI-PING, ZHU SHI-ZHENG, JIANG XI-KUI, LI ZHAN-TING: "F ... H-N hydrogen bonding driven foldamers: efficient receptors for dialkylammonium ions", ANGEWANDTE CHEMIE, vol. 44, no. 35, 2005, pages 5725 - 5729, XP055773480
DATABASE REGISTRY [online] 29 March 2004 (2004-03-29), "CN -1,3-Benzenedicarboxamide, 2-fluoro-N1,N3-bis(4-fluorophenyl)-(CA INDEX NAME)", XP055773824, retrieved from STN Database accession no. 668468-70-0
HABA OSAMU, SEINO HIROSHI, AOKI KAZUTAKA, IGUCHI KAZUYUKI, UEDA MITSURU: "Synthesis of ordered polymer by direct polycondensation. VIII. Ordered polymer from two nonsymmetric monomers", JOURNAL OF POLYMER SCIENCE , PART A: POLYMER CHEMISTRY, vol. 36, no. 13, 1998, pages 2309 - 2314, XP055773485
DATABASE REGISTRY [online] 29 March 2004 (2004-03-29), "CN -1,3-Benzenedicarboxamide, N1,N3-bis(4-chlorophenyl)-2-fluoro-(CA INDEX NAME)", XP055773835, retrieved from STN Database accession no. 668468-69-7
SELZER LISA, KATEN SARAH P., ZLOTNICK ADAM: "The Hepatitis B Virus Core Protein Intradimer Interface Modulates Capsid Assembly and Stability", BIOCHEMISTRY, vol. 53, no. 34, 2014, pages 5496 - 5504, XP055773492
Attorney, Agent or Firm:
IKEUCHI & PARTNERS (JP)
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