Title:
CANNABINOID RECEPTOR MODULATOR
Document Type and Number:
WIPO Patent Application WO/2005/000829
Kind Code:
A1
Abstract:
A cannabinoid receptor modulator which contains a compound represented by the formula (I0): (I0) (wherein X represents oxygen, etc.; R0 represents optionally substituted acylamino; ring A0 represents a benzene ring optionally having a substituent besides R0; and ring B represents optionally substituted five-membered heterocycle), a salt of the compound, or a prodrug of either.
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Inventors:
OHKAWA SHIGENORI (JP)
TSUKAMOTO TETSUYA (JP)
KIYOTA YOSHIHIRO (JP)
GOTO MIKA (JP)
YAMAMOTO SHOUZOU (JP)
SHIMOJOU MASATO (JP)
SETOU MASAKI (JP)
TSUKAMOTO TETSUYA (JP)
KIYOTA YOSHIHIRO (JP)
GOTO MIKA (JP)
YAMAMOTO SHOUZOU (JP)
SHIMOJOU MASATO (JP)
SETOU MASAKI (JP)
Application Number:
PCT/JP2004/009355
Publication Date:
January 06, 2005
Filing Date:
June 25, 2004
Export Citation:
Assignee:
TAKEDA PHARMACEUTICAL (JP)
OHKAWA SHIGENORI (JP)
TSUKAMOTO TETSUYA (JP)
KIYOTA YOSHIHIRO (JP)
GOTO MIKA (JP)
YAMAMOTO SHOUZOU (JP)
SHIMOJOU MASATO (JP)
SETOU MASAKI (JP)
OHKAWA SHIGENORI (JP)
TSUKAMOTO TETSUYA (JP)
KIYOTA YOSHIHIRO (JP)
GOTO MIKA (JP)
YAMAMOTO SHOUZOU (JP)
SHIMOJOU MASATO (JP)
SETOU MASAKI (JP)
International Classes:
A61K31/343; A61K31/357; A61K31/381; A61K31/4025; A61K31/4178; A61K31/426; A61K31/443; A61K31/453; A61K31/506; A61P3/04; A61P11/06; A61P25/00; A61P25/08; A61P27/06; A61P43/00; C07D307/86; C07D333/54; (IPC1-7): C07D307/79; C07D307/80; C07D405/10; C07D333/54; C07D405/06; C07D407/04; C07D405/04; C07D417/04; C07D409/04; A61K31/343; A61K31/4025; A61K31/357; A61K31/443; A61K31/506; A61K31/426; A61K31/381; A61K31/4178; A61K31/453; A61P3/04; A61P11/06; A61P25/00; A61P25/08; A61P27/06; A61P43/00
Domestic Patent References:
| WO2000034262A1 | 2000-06-15 |
Foreign References:
| JPH11503467A | 1999-03-26 | |||
| JPH10330380A | 1998-12-15 | |||
| JPH10505089A | 1998-05-19 | |||
| JP2002348239A | 2002-12-04 | |||
| JPH05140142A | 1993-06-08 | |||
| JPH11500411A | 1999-01-12 | |||
| JPH10503185A | 1998-03-24 |
Other References:
OHKAWA S. ET AL: "5-Aminocoumarans: Dual Inhibitors of Lipid Peroxidation and Dopamine Release with Protective Effects against Central Nervous System Trauma and Ischemia", JOURNAL OF MEDICINAL CHEMISTRY, vol. 40, no. 4, 1997, pages 559 - 573, XP002979756
JANUSZ J.M: ET AL: "New Cyclooxygenase-2/5-Lipoxygenase Inhibitors. 3. 7-tert-Butyl-2,3- dihydro-3,3-dimethylbenzofuran Derivatives as Gastrointestinal Safe Antiinflammatory and Analgesic Agents: Variations at the 5 Position", JOURNAL OF MEDICINAL CHEMISTRY, vol. 41, no. 18, 1998, pages 3515 - 3529, XP002223203
"Mitsunobu reaction", SYNTHESIS, 1981, pages 1 - 27
See also references of EP 1637527A4
JANUSZ J.M: ET AL: "New Cyclooxygenase-2/5-Lipoxygenase Inhibitors. 3. 7-tert-Butyl-2,3- dihydro-3,3-dimethylbenzofuran Derivatives as Gastrointestinal Safe Antiinflammatory and Analgesic Agents: Variations at the 5 Position", JOURNAL OF MEDICINAL CHEMISTRY, vol. 41, no. 18, 1998, pages 3515 - 3529, XP002223203
"Mitsunobu reaction", SYNTHESIS, 1981, pages 1 - 27
See also references of EP 1637527A4
Attorney, Agent or Firm:
Kawamiya, Osamu (IMP Building 3-7, Shiromi 1-chome, Chuo-k, Osaka-shi Osaka 01, JP)
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