CRYSTAL OF BICYCLIC FUSED HETEROCYCLIC DERIVATIVE, PROCESS FOR PRODUCTION THEREOF, AND USE THEREOF

Title:

CRYSTAL OF BICYCLIC FUSED HETEROCYCLIC DERIVATIVE, PROCESS FOR PRODUCTION THEREOF, AND USE THEREOF

Document Type and Number:

WIPO Patent Application WO/2006/070934

Kind Code:

A1

Abstract:

A crystal of a p-toluenesulphonate salt of 5-(5-[[2-(2-chlorophenyl)ethyl]amino]pentanoyl)-1,3- dimethyl-1,3-dihydro-2H-benzoimidazol-2-one, a pharmaceutical composition comprising the crystal, a process for producing the crystal, and use of the crystal. The crystal has excellent acetylcholinesterase inhibitory activity and effects of preventing and/or treating dysuria and also has excellent stability.

More Like This:

JP2009527525	Benzoimidazolone derivative for the treatment of urinary incontinence
WO/2007/048842	BENZIMIDAZOLE DERIVATIVES FOR USE AS BETA-3 RECEPTOR AGONISTS

Inventors:

KIMURA KAZUHIRO (JP)
KORO NORIAKI (JP)
YAMASAKI SEIJI (JP)

Application Number:

PCT/JP2005/024260

Publication Date:

July 06, 2006

Filing Date:

December 28, 2005

Export Citation:

Click for automatic bibliography generation Help

Assignee:

TAKEDA PHARMACEUTICAL (JP)
KIMURA KAZUHIRO (JP)
KORO NORIAKI (JP)
YAMASAKI SEIJI (JP)

International Classes:

C07D235/26; A61K31/4184; A61P7/10; A61P13/10; A61P43/00

Foreign References:

JP2003335701A	2003-11-28
JP2005035996A	2005-02-10

Attorney, Agent or Firm:

Takashima, Hajime (1-1 Fushimimachi 4-chome, Chuo-ku, Osaka-sh, Osaka 44, JP)

Download PDF:

View/Download PDF PDF Help

Previous Patent: PYRIMIDINYLISOXAZOL DERIVATIVE

Next Patent: ELECTROSTATIC COATER