Title:
CRYSTALLINE PHASES OF 2'-{[2-(4-METHOXY-PHENYL)-ACETYLAMINO]-METHYL}-BIPHENYL-2-CARBOXYLIC ACID (2-PYRIDIN-3-YL-ETHYL)-AMIDE
Document Type and Number:
WIPO Patent Application WO/2010/139585
Kind Code:
A3
Abstract:
The present invention relates to polymorphic forms and solvates of 2'-{[2-(4-methoxy-phenyl)-acetylamino]-methyl]}-biphenyl-2-carboxylic acid (2-pyhdin-3-yl-ethyl)-amide, processes for their preparation and their use, in particular for the preparation of medicaments.
Inventors:
NAGEL NORBERT (DE)
BERCHTOLD HARALD (DE)
SCHUR MICHAEL (DE)
HOERSTERMANN DIRK (DE)
BERCHTOLD HARALD (DE)
SCHUR MICHAEL (DE)
HOERSTERMANN DIRK (DE)
Application Number:
PCT/EP2010/057273
Publication Date:
May 05, 2011
Filing Date:
May 26, 2010
Export Citation:
Assignee:
SANOFI AVENTIS DEUTSCHLAND (DE)
NAGEL NORBERT (DE)
BERCHTOLD HARALD (DE)
SCHUR MICHAEL (DE)
HOERSTERMANN DIRK (DE)
NAGEL NORBERT (DE)
BERCHTOLD HARALD (DE)
SCHUR MICHAEL (DE)
HOERSTERMANN DIRK (DE)
International Classes:
A61K31/4406; C07D213/16
Foreign References:
US20070043091A1 | 2007-02-22 | |||
US6531495B1 | 2003-03-11 |
Other References:
CAIRA M R: "CRYSTALLINE POLYMORPHISM OF ORGANIC COMPOUNDS", TOPICS IN CURRENT CHEMISTRY, SPRINGER, BERLIN, DE, vol. 198, 1 January 1998 (1998-01-01), pages 163 - 208, XP001156954
Attorney, Agent or Firm:
MICHALSKI HÜTTERMANN & PARTNER PATENTANWÄLTE (Düsseldorf, DE)
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