Title:
DIARYL ETHERS AS OPIOID RECEPTOR ANTAGONIST
Document Type and Number:
WIPO Patent Application WO2004026305
Kind Code:
A9
Abstract:
A compound of the formula (I) wherein the variables X1 to X10, R<1> to R<7> including R<3'>, E, v, y, z, A and B are as described, or a pharmaceutically acceptable salt, solvate, enantiomer, racemate, diastereomer or mixtures thereof, useful for the treatment, prevention or amelioration of obesity and Related Diseases is disclosed.
Inventors:
BLANCO-PILLADO MARIA-JESUS (US)
CHAPPELL MARK DONALD (US)
DE LA TORRE MARTA GARCIA (ES)
DIAZ BUEZO NURIA (ES)
FRITZ JAMES ERWIN (US)
HOLLOWAY WILLIAM GLEN (US)
MATT JAMES EDWARD JUNIOR (US)
MITCH CHARLES HOWARD (US)
PEDREGAL-TERCERO CONCEPCION (ES)
QUIMBY STEVEN JAMES (US)
SIEGEL MILES GOODMAN (US)
SMITH DANA RAE (US)
STUCKY RUSSELL DEAN (US)
TAKEUCHI KUMIKO (US)
THOMAS ELIZABETH MARIE (US)
WOLFE CHAD NOLAN (US)
CHAPPELL MARK DONALD (US)
DE LA TORRE MARTA GARCIA (ES)
DIAZ BUEZO NURIA (ES)
FRITZ JAMES ERWIN (US)
HOLLOWAY WILLIAM GLEN (US)
MATT JAMES EDWARD JUNIOR (US)
MITCH CHARLES HOWARD (US)
PEDREGAL-TERCERO CONCEPCION (ES)
QUIMBY STEVEN JAMES (US)
SIEGEL MILES GOODMAN (US)
SMITH DANA RAE (US)
STUCKY RUSSELL DEAN (US)
TAKEUCHI KUMIKO (US)
THOMAS ELIZABETH MARIE (US)
WOLFE CHAD NOLAN (US)
Application Number:
PCT/US2003/026300
Publication Date:
May 13, 2004
Filing Date:
September 17, 2003
Export Citation:
Assignee:
LILLY CO ELI (US)
BLANCO-PILLADO MARIA-JESUS (US)
CHAPPELL MARK DONALD (US)
DE LA TORRE MARTA GARCIA (ES)
DIAZ BUEZO NURIA (ES)
FRITZ JAMES ERWIN (US)
HOLLOWAY WILLIAM GLEN (US)
MATT JAMES EDWARD JUNIOR (US)
MITCH CHARLES HOWARD (US)
PEDREGAL-TERCERO CONCEPCION (ES)
QUIMBY STEVEN JAMES (US)
SIEGEL MILES GOODMAN (US)
SMITH DANA RAE (US)
STUCKY RUSSELL DEAN (US)
TAKEUCHI KUMIKO (US)
THOMAS ELIZABETH MARIE (US)
WOLFE CHAD NOLAN (US)
BLANCO-PILLADO MARIA-JESUS (US)
CHAPPELL MARK DONALD (US)
DE LA TORRE MARTA GARCIA (ES)
DIAZ BUEZO NURIA (ES)
FRITZ JAMES ERWIN (US)
HOLLOWAY WILLIAM GLEN (US)
MATT JAMES EDWARD JUNIOR (US)
MITCH CHARLES HOWARD (US)
PEDREGAL-TERCERO CONCEPCION (ES)
QUIMBY STEVEN JAMES (US)
SIEGEL MILES GOODMAN (US)
SMITH DANA RAE (US)
STUCKY RUSSELL DEAN (US)
TAKEUCHI KUMIKO (US)
THOMAS ELIZABETH MARIE (US)
WOLFE CHAD NOLAN (US)
International Classes:
A61P3/04; C07C235/46; C07D213/38; C07D213/643; C07D213/78; C07D213/81; C07D213/82; C07D217/04; C07D237/24; C07D241/24; C07D307/14; C07D333/20; C07D401/06; C07D401/12; C07D401/14; C07D405/12; C07D409/12; C07D409/14; C07D413/12; C07D417/12; C07D417/14; C07D213/64; (IPC1-7): A61K31/4412; C07D213/82; C07D401/12; C07D241/24; C07D401/06; C07D333/20; A61K31/4427; A61P3/04; C07C43/20
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