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Title:
FUSED HETEROCYCLIC COMPOUNDS AND ANALOGS THEREOF: MODULATORS OF NUCLEAR HORMONE RECEPTOR FUNCTION
Document Type and Number:
WIPO Patent Application WO2003053358
Kind Code:
A3
Abstract:
Fused cyclic compounds, methods of using such compounds in the treatment of nuclear hormone receptor-associated conditions such as cancer and immune disorders, and pharmaceutical compositions containing such compounds.

Inventors:
SALVATI MARK E (US)
BALOG JAMES AARON (US)
PICKERING DACIA A (US)
ZHU HONG (US)
Application Number:
PCT/US2002/040737
Publication Date:
October 02, 2003
Filing Date:
December 18, 2002
Export Citation:
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Assignee:
BRISTOL MYERS SQUIBB CO (US)
SALVATI MARK E (US)
BALOG JAMES AARON (US)
PICKERING DACIA A (US)
ZHU HONG (US)
International Classes:
A61K31/403; C07D231/56; A61K31/407; A61K31/416; A61K31/428; A61K31/4709; A61K45/00; A61P3/06; A61P3/10; A61P5/26; A61P9/00; A61P9/02; A61P13/08; A61P15/00; A61P15/12; A61P15/18; A61P17/00; A61P17/14; A61P19/10; A61P25/18; A61P25/28; A61P25/36; A61P35/00; A61P37/00; A61P43/00; C07B61/00; C07D209/72; C07D209/74; C07D209/76; C07D231/54; C07D275/06; C07D401/04; C07D491/18; C07D513/18; (IPC1-7): C07D275/06
Other References:
BEER ET AL.: "Studies of 5-benzoyl-3-isothiazolinones", TETRAHEDRON, vol. 37, no. 22, 1981, pages 3867 - 3870, XP002964123
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