Title:
GPR14 ANTAGONIST
Document Type and Number:
WIPO Patent Application WO/2002/002530
Kind Code:
A1
Abstract:
A novel GPR14 antagonist. The GPR14 antagonist comprises a compound represented by the formula (I) or a salt thereof wherein Ar represents optionally substituted aryl; X represents a spacer; n is an integer of 1 to 10; R represents an optionally substituted hydrocarbon group, etc., provided that R may be bonded to Ar, etc. to form a ring; and Y represents optionally substituted amino, etc.
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Inventors:
TARUI NAOKI (JP)
SANTO TAKASHI (JP)
WATANABE HIROYUKI (JP)
ASO KAZUYOSHI (JP)
ISHIHARA YUJI (JP)
SANTO TAKASHI (JP)
WATANABE HIROYUKI (JP)
ASO KAZUYOSHI (JP)
ISHIHARA YUJI (JP)
Application Number:
PCT/JP2001/005784
Publication Date:
January 10, 2002
Filing Date:
July 04, 2001
Export Citation:
Assignee:
TAKEDA CHEMICAL INDUSTRIES LTD (JP)
TARUI NAOKI (JP)
SANTO TAKASHI (JP)
WATANABE HIROYUKI (JP)
ASO KAZUYOSHI (JP)
ISHIHARA YUJI (JP)
TARUI NAOKI (JP)
SANTO TAKASHI (JP)
WATANABE HIROYUKI (JP)
ASO KAZUYOSHI (JP)
ISHIHARA YUJI (JP)
International Classes:
A61P9/08; A61P9/10; A61P9/12; A61P43/00; C07D223/16; (IPC1-7): C07D223/16; A61K31/55; A61P9/08; A61P9/10; A61P9/12; A61P43/00; C07D401/12; C07D405/12; C07D413/12
Domestic Patent References:
WO1998046590A1 | 1998-10-22 | |||
WO2000023437A1 | 2000-04-27 | |||
WO2000032627A1 | 2000-06-08 |
Foreign References:
EP0560235A1 | 1993-09-15 | |||
EP0487071A1 | 1992-05-27 |
Other References:
See also references of EP 1310490A4
Attorney, Agent or Firm:
Aoyama, Tamotsu (Shiromi 1-chome Chuo-ku Osaka |shi, Osaka, JP)
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