Title:
HETEROARYL 5-THIO-β-D-GLUCOPYRANOSIDE DERIVATIVES AND REMEDIES FOR DIABETES CONTAINING THE SAME
Document Type and Number:
WIPO Patent Application WO/2004/089967
Kind Code:
A1
Abstract:
It is intended to provide heteroaryl 5-thio-β-D-glucopyranoside compounds represented by the following general formula which show an effect of inhibiting the activity of SGLT2, pharmaceutically acceptable salts thereof or hydrates of the same; and drugs containing the same as the active ingredient, in particular, remedies for diabetes, diabetes-related diseases or complications of diabetes.
Inventors:
KAKINUMA HIROYUKI (JP)
SATO MASAKAZU (JP)
AMADA HIDEAKI (JP)
ASANUMA HAJIME (JP)
TSUCHIYA YUKO (JP)
SATO MASAKAZU (JP)
AMADA HIDEAKI (JP)
ASANUMA HAJIME (JP)
TSUCHIYA YUKO (JP)
Application Number:
PCT/JP2004/001272
Publication Date:
October 21, 2004
Filing Date:
February 06, 2004
Export Citation:
Assignee:
TAISHO PHARMACEUTICAL CO LTD (JP)
KAKINUMA HIROYUKI (JP)
SATO MASAKAZU (JP)
AMADA HIDEAKI (JP)
ASANUMA HAJIME (JP)
TSUCHIYA YUKO (JP)
KAKINUMA HIROYUKI (JP)
SATO MASAKAZU (JP)
AMADA HIDEAKI (JP)
ASANUMA HAJIME (JP)
TSUCHIYA YUKO (JP)
International Classes:
A61K31/7056; A61K31/706; A61P3/10; A61P43/00; C07H17/00; C07H17/02; (IPC1-7): C07H17/02; A61K31/7056; A61P3/10; A61P43/00
Domestic Patent References:
| WO2002068440A1 | 2002-09-06 | |||
| WO2001016147A1 | 2001-03-08 | |||
| WO2002036602A1 | 2002-05-10 |
Other References:
SAKAGUCHI M. ET AL: "Potential Radiosensitizing Agents 4. 2-Nitroimidazole Nucleosides", J. MED. CHEM., vol. 25, no. 11, 1982, pages 1339 - 1342, XP002979334
See also references of EP 1609799A4
See also references of EP 1609799A4
Attorney, Agent or Firm:
Shamoto, Ichio (Section 206 New Ohtemachi Bldg., 2-1,
Ohtemachi 2-chom, Chiyoda-ku Tokyo 04, JP)
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