Title:
HETEROARYL AMIDE COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITIONS THEREOF, AND APPLICATIONS THEREOF
Document Type and Number:
WIPO Patent Application WO/2019/085978
Kind Code:
A1
Abstract:
The present invention relates to heteroaryl amide compounds, a preparation method therefor, pharmaceutical compositions thereof and applications thereof, and specifically, relates to a type of compounds having broad-spectrum tumor resistant activity, a preparation method therefor, pharmaceutical compositions containing the compounds, and uses of the compounds in the preparation of drugs for treating tumors.
Inventors:
REN RUIBAO (CN)
DENG XIANMING (CN)
WU MIN (CN)
ZHANG TING (CN)
JIAO BO (CN)
KANG QIAOFENG (CN)
HUANG WEI (CN)
DENG XIANMING (CN)
WU MIN (CN)
ZHANG TING (CN)
JIAO BO (CN)
KANG QIAOFENG (CN)
HUANG WEI (CN)
Application Number:
PCT/CN2018/113549
Publication Date:
May 09, 2019
Filing Date:
November 02, 2018
Export Citation:
Assignee:
RUI JIN HOSPITAL AFFILIATED TO SHANGHAI JIAO TONG UNIV SCHOOL OF MEDICINE (CN)
UNIV XIAMEN (CN)
UNIV XIAMEN (CN)
International Classes:
C07D513/04; A61K31/425; A61P35/00
Foreign References:
| CN101790313A | 2010-07-28 |
Other References:
SARTORI, LUCA ET AL.: "Thieno[3, 2-b]pyrrole-5-carboxamides as New Rever- sible Inhibitors of Histone Lysine Demethylase KDMIA/LSDI.Part 1.High-Throu- ghput Screening and reliminary Exploration", JOURNAL OF MEDICINAL CHEMISTRY, vol. 60, no. 5, 10 February 2017 (2017-02-10), pages 1673 - 1692, XP055507204
"Burger's Medicinal Chemistry and Drug Discovery", 1995, MACK PUBLISHING COMPANY, pages: 172 - 178,949-982
"Purification of Laboratory Chemicals", 1980, D. R.; PERGAMON PRESS
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 87, 2014, pages 529 - 539
See also references of EP 3705481A4
"Burger's Medicinal Chemistry and Drug Discovery", 1995, MACK PUBLISHING COMPANY, pages: 172 - 178,949-982
"Purification of Laboratory Chemicals", 1980, D. R.; PERGAMON PRESS
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 87, 2014, pages 529 - 539
See also references of EP 3705481A4
Attorney, Agent or Firm:
CCPIT PATENT AND TRADEMARK LAW OFFICE (CN)
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