Title:
HETEROCYCLIC COMPOUND AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2011/002067
Kind Code:
A1
Abstract:
Disclosed are a heterocyclic derivative which has excellent amyloid β production inhibitory activity, and a use of the heterocyclic derivative.
Specifically disclosed is a compound represented by formula (I) or a salt thereof.
(In the formula, the symbols are as defined in the description.)
Inventors:
TERAUCHI JUN (JP)
KOIKE TATSUKI (JP)
HONDA EIJI (JP)
NAKAMURA MINORU (JP)
KAJITA YUICHI (JP)
HOASHI YASUTAKA (JP)
MORIMOTO SACHIE (JP)
FUJIMOTO TATSUHIKO (JP)
KOIKE TATSUKI (JP)
HONDA EIJI (JP)
NAKAMURA MINORU (JP)
KAJITA YUICHI (JP)
HOASHI YASUTAKA (JP)
MORIMOTO SACHIE (JP)
FUJIMOTO TATSUHIKO (JP)
Application Number:
PCT/JP2010/061280
Publication Date:
January 06, 2011
Filing Date:
July 01, 2010
Export Citation:
Assignee:
TAKEDA PHARMACEUTICAL (JP)
TERAUCHI JUN (JP)
KOIKE TATSUKI (JP)
HONDA EIJI (JP)
NAKAMURA MINORU (JP)
KAJITA YUICHI (JP)
HOASHI YASUTAKA (JP)
MORIMOTO SACHIE (JP)
FUJIMOTO TATSUHIKO (JP)
TERAUCHI JUN (JP)
KOIKE TATSUKI (JP)
HONDA EIJI (JP)
NAKAMURA MINORU (JP)
KAJITA YUICHI (JP)
HOASHI YASUTAKA (JP)
MORIMOTO SACHIE (JP)
FUJIMOTO TATSUHIKO (JP)
International Classes:
C07D231/12; A61K31/439; A61K31/496; A61K31/506; A61K31/5377; A61K31/541; A61K31/551; A61P25/28; A61P43/00; C07D249/06; C07D249/08; C07D261/08; C07D263/32; C07D271/06; C07D271/10; C07D277/28; C07D333/20; C07D401/12; C07D403/04; C07D403/10; C07D403/12; C07D403/14; C07D405/12; C07D409/12; C07D413/10; C07D413/12; C07D413/14; C07D417/12; C07D417/14; C07D471/04; C07D471/08; C07D487/08; C07D491/107; C07D498/08
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Other References:
RAKESH ET AL.: "Synthesis, optimization and structure-activity relationships of 3,5-disubstituted isoxazolines as new anti-tuberculosis agents", EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 44, no. 2, 2009, pages 460 - 472, XP025950175, DOI: doi:10.1016/j.ejmech.2008.04.007
Attorney, Agent or Firm:
TAKASHIMA, HAJIME (JP)
Takashima 1 (JP)
Takashima 1 (JP)
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