MEDICINAL COMPOSITIONS OF NONPEPTIDYL GONADOTROPIN-RELEASING HORMONE AGONIST OR ANTAGONIST, PROCESS FOR PRODUCING THE SAME AND USE THEREOF

WIPO Patent Application WO/2002/047722

A1

Medicinal compositions comprising: (i) a nonpeptidyl gonadotropin-releasing hormone agonist or antagonist; (ii) an organic acid or its salt; and (iii) a biodegradable polymer or its salt. These compositions can be efficiently produced, suffer from no trouble in quality control and can achieve a stable releasing speed over a long period of time, even in case where the nonpeptidyl GnRH agonist or antagonist is contained in a large amount regardless of the solubility, melting point or crystallinity thereof.

SUZUKI HIROSHI (JP)
HATA YOSHIO (JP)

PCT/JP2001/010956

June 20, 2002

December 14, 2001

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TAKEDA CHEMICAL INDUSTRIES LTD (JP)
SUZUKI HIROSHI (JP)
HATA YOSHIO (JP)

A61K9/52; A61K31/00; A61K31/4365; A61K31/519; A61K47/12; A61K47/34; A61P1/00; A61P5/24; A61P13/08; A61P15/00; A61P15/08; A61P15/18; A61P17/00; A61P17/14; A61P25/28; A61P35/04; C07D333/38; C07D471/04; C07D487/04; C07D495/04; (IPC1-7): A61K45/00; A61K9/50; A61K9/52; A61K31/4365; A61K31/519; A61K47/12; A61K47/34; A61P1/00; A61P5/24; A61P13/08; A61P15/00; A61P15/08; A61P15/18; A61P17/00; A61P17/14; A61P25/28; A61P35/04; A61P34/00

WO1999036099A1	1999-07-22
WO1998032423A1	1998-07-30
WO1995015767A1	1995-06-15
WO1995028405A1	1995-10-26
WO1996024597A1	1996-08-15
WO2000056739A1	2000-09-28

EP0626170A2	1994-11-30
JP2001081043A	2001-03-27

Aoyama, Tamotsu (Shiromi 1-chome Chuo-ku Osaka-shi, Osaka, JP)

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