Title:
METHOD FOR PREPARING IBRUTINIB
Document Type and Number:
WIPO Patent Application WO/2016/127915
Kind Code:
A1
Abstract:
The present application relates to a method for preparing Ibrutinib as shown by the following synthetic route and the intermediate compounds involved therein.
Inventors:
ZHANG XIQUAN (CN)
KONG RUI (CN)
LIU XIN (CN)
CHEN SHAN (CN)
CHEN XIAOPING (CN)
YANG LEILEI (CN)
ZHANG AIMING (CN)
CHENG XINGDONG (CN)
KONG RUI (CN)
LIU XIN (CN)
CHEN SHAN (CN)
CHEN XIAOPING (CN)
YANG LEILEI (CN)
ZHANG AIMING (CN)
CHENG XINGDONG (CN)
Application Number:
PCT/CN2016/073537
Publication Date:
August 18, 2016
Filing Date:
February 04, 2016
Export Citation:
Assignee:
SHANGHAI DUDE MEDICAL SCIENCE AND TECH CO LTD (CN)
CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD (CN)
LIANYUNGANG RUNZHONG PHARMACEUTICAL CO LTD (CN)
CHIA TAI TIANQING PHARMACEUTICAL GROUP CO LTD (CN)
LIANYUNGANG RUNZHONG PHARMACEUTICAL CO LTD (CN)
International Classes:
C07D487/04
Foreign References:
CN101610676A | 2009-12-23 | |||
CN103121999A | 2013-05-29 | |||
CN105017256A | 2015-11-04 |
Other References:
See also references of EP 3257855A4
Attorney, Agent or Firm:
INSIGHT INTELLECTUAL PROPERTY LIMITED (CN)
北京英赛嘉华知识产权代理有限责任公司 (CN)
北京英赛嘉华知识产权代理有限责任公司 (CN)
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