MONO- AND DISUBSTITUTED 3-PROPYL GAMMA-AMINOBUTYRIC ACIDS

WIPO Patent Application WO2000076958

A3

The instant invention is a series of novel mono- and disubstituted 3-propyl gamma aminobutyric acids of Formula (I). The compounds are useful as therapeutic agents in the treatment of epilepsy, faintness attacks, hypokinesia, cranial disorders, neurodegenerative disorders, depression, anxiety, panic, pain, neuropathological disorders, arthritis, sleep disorders, IBS, and gastric damage. Methods of preparing the compounds and useful intermediates are also part of the invention.

BELLIOTTI THOMAS RICHARD (US)
BRYANS JUSTIN STEPHEN (GB)
EKHATO IHOEZO VICTOR (US)
OSUMA AUGUSTINE TOBI (US)
SCHELKUN ROBERT MICHAEL (US)
THORPE ANDREW JOHN (US)
WISE LAWRENCE DAVID (US)
WUSTROW DAVID JUERGEN (US)
YUEN PO-WAI (US)
SCHWARZ JACOB BRADLEY (US)

PCT/US2000/015070

April 12, 2001

May 31, 2000

Click for automatic bibliography generation  

WARNER LAMBERT CO (US)
BELLIOTTI THOMAS RICHARD (US)
BRYANS JUSTIN STEPHEN (GB)
EKHATO IHOEZO VICTOR (US)
OSUMA AUGUSTINE TOBI (US)
SCHELKUN ROBERT MICHAEL (US)
THORPE ANDREW JOHN (US)
WISE LAWRENCE DAVID (US)
WUSTROW DAVID JUERGEN (US)
YUEN WAI (US)
SCHWARZ JACOB BRADLEY (US)

A61K31/197; A61P1/00; A61P25/00; A61P25/08; A61P25/10; A61P25/20; A61P25/22; A61P25/24; A61P29/02; A61P43/00; C07C229/08; C07C229/20; C07C229/22; C07C229/28; C07C229/30; C07C229/32; C07C229/34; C07C229/36; A61K; A61P; C07C; (IPC1-7): C07C229/08; A61K31/197; C07C229/30; C07C229/22; C07C229/34; C07C229/32; C07C229/20; A61P25/00; A61P1/00

WO1992009560A1	1992-06-11
WO1998017627A1	1998-04-30
WO1999021824A1	1999-05-06

View/Download PDF      PDF Help

Previous Patent: ENANTIOMERS OF N-DESMETHYL VENLAFAXINE

Next Patent: INTERMEDIATES FOR THE PREPARATION OF (N)-[2-(CARBOXYMETHOXY) ETHYL]-(N)-(CARBOXYMETHYL) GLYCINE