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Title:
NITROGEN-CONTAINING TRICYCLIC DERIVATIVE HAVING HIV REPLICATION INHIBITORY ACTIVITY
Document Type and Number:
WIPO Patent Application WO/2016/194806
Kind Code:
A1
Abstract:
Provided are: a novel compound having antiviral action, especially HIV replication inhibitory activity; and a pharmaceutical product, especially an anti-HIV agent which contains this compound. A compound represented by formula (I). (In the formula, A3 represents CR3A, CR3AR3B, N or NR3C; each of R3A, R3B, R4A and R4B independently represents a hydrogen atom, a halogen atom, a cyano group, a substituted or unsubstituted alkyl group, a substituted or unsubstituted alkynyl group or a substituted or unsubstituted non-aromatic carbocyclic group; R3C represents a hydrogen atom, a substituted or unsubstituted alkyl group or a substituted or unsubstituted non-aromatic carbocyclic group; ring T1 represents a substituted or unsubstituted nitrogen-containing non-aromatic heterocyclic ring; R1 represents a hydrogen atom, a halogen atom, a cyano group or a substituted or unsubstituted alkyl group; each R2 independently represents a substituted or unsubstituted alkyl group or the like; n represents 1 or 2; R3 represents a substituted or unsubstituted aromatic carbocyclic group or the like; and R4 represents a hydrogen atom or a carboxy-protecting group.)

Inventors:
TAMURA YOSHINORI (JP)
KAWASUJI TAKASHI (JP)
SUGIYAMA SHUICHI (JP)
MATSUMURA AKIRA (JP)
AKIYAMA TOSHIYUKI (JP)
TOMIDA YUTAKA (JP)
Application Number:
PCT/JP2016/065702
Publication Date:
December 08, 2016
Filing Date:
May 27, 2016
Export Citation:
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Assignee:
SHIONOGI & CO (JP)
International Classes:
C07D487/06; A61K31/4985; A61K31/554; A61P31/12; A61P31/18; C07D513/06
Domestic Patent References:
WO2014119636A12014-08-07
WO2015174511A12015-11-19
WO2015147247A12015-10-01
Foreign References:
JP2009503069A2009-01-29
JP2013535426A2013-09-12
JP2014511872A2014-05-19
JP2012526728A2012-11-01
JP2005516031A2005-06-02
JP2003510324A2003-03-18
JP2000505450A2000-05-09
JP2004256531A2004-09-16
Other References:
See also references of EP 3305789A4
Attorney, Agent or Firm:
YAMAUCHI, Hideaki et al. (JP)
Hideaki Yamauchi (JP)
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