Title:
NOVEL AZETIDINE DERIVATIVE OR SALT THEREOF
Document Type and Number:
WIPO Patent Application WO/2004/007446
Kind Code:
A1
Abstract:
A compound represented by the following formula (I), which has excellent dipeptidyl peptidase IV inhibitory activity; and a therapeutic agent which, based on the activity, is highly effective against insulin dependent diabetes (type 1 diabetes), especially noninsulin-dependent diabetes (type 2 diabetes), insulin-resistant diseases, and obesity. (I) (The substituents are as defined in claim 1.)
Inventors:
HAYAKAWA MASAHIKO (JP)
NEGORO KENJI (JP)
SUZUKI TAKAYUKI (JP)
MARUYAMA TATSUYA (JP)
NAKANO RYOSUKE (JP)
NEGORO KENJI (JP)
SUZUKI TAKAYUKI (JP)
MARUYAMA TATSUYA (JP)
NAKANO RYOSUKE (JP)
Application Number:
PCT/JP2003/008727
Publication Date:
January 22, 2004
Filing Date:
July 09, 2003
Export Citation:
Assignee:
YAMANOUCHI PHARMA CO LTD (JP)
HAYAKAWA MASAHIKO (JP)
NEGORO KENJI (JP)
SUZUKI TAKAYUKI (JP)
MARUYAMA TATSUYA (JP)
NAKANO RYOSUKE (JP)
HAYAKAWA MASAHIKO (JP)
NEGORO KENJI (JP)
SUZUKI TAKAYUKI (JP)
MARUYAMA TATSUYA (JP)
NAKANO RYOSUKE (JP)
International Classes:
A61P3/04; A61P3/10; A61P43/00; C07D205/04; (IPC1-7): C07D205/04; A61K31/397; A61K31/439; A61K31/4427; A61K31/4439; A61K31/4523; A61K31/4725; A61K31/497; A61K31/506; A61P3/04; A61P3/10; A61P43/00; C07D401/06; C07D401/12; C07D401/14; C07D453/02
Domestic Patent References:
| WO2003057666A2 | 2003-07-17 | |||
| WO2003057144A2 | 2003-07-17 | |||
| WO2002038541A1 | 2002-05-16 | |||
| WO2002030890A1 | 2002-04-18 | |||
| WO2001096295A2 | 2001-12-20 | |||
| WO2001062266A2 | 2001-08-30 | |||
| WO2000034241A1 | 2000-06-15 | |||
| WO1998019998A2 | 1998-05-14 |
Attorney, Agent or Firm:
Nagai, Shozo c/o Yamanouchi Pharmaceutical Co. Ltd. (Patent Department, 17-1, Hasune 3-chom, Itabashi-ku Tokyo, JP)
Download PDF: