NOVEL PYRIDYL BENZOXAZINE DERIVATIVES, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AND USE THEREOF

Title:

NOVEL PYRIDYL BENZOXAZINE DERIVATIVES, PHARMACEUTICAL COMPOSITION COMPRISING THE SAME, AND USE THEREOF

Document Type and Number:

WIPO Patent Application WO/2012/050380

Kind Code:

A2

Abstract:

Discloses is a benzoxazine benzimidazole derivative, represented by Chemical Formula 1, functioning as an antagonist to the vanilloid receptor-1, a pharmaceutical composition comprising the same, and the use thereof. The benzoxazine benzimidazole derivative can be useful for preventing or treating a disease associated with antagonistic activity of vanilloid receptor-1, without hyperthermia.

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Inventors:

KIM JI DUCK (KR)
YOON HONG CHUL (KR)
KIM IN WOO (KR)
CHO MIN JAE (KR)
LEE IN YOUNG (KR)
LEE SANG HO (KR)
PARK EUN KYUNG (KR)
LIM KWON JO (KR)
NAM SANG HYUN (KR)

Application Number:

PCT/KR2011/007635

Publication Date:

April 19, 2012

Filing Date:

October 13, 2011

Export Citation:

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Assignee:

DAE WOONG PHARMA (KR)
KIM JI DUCK (KR)
YOON HONG CHUL (KR)
KIM IN WOO (KR)
CHO MIN JAE (KR)
LEE IN YOUNG (KR)
LEE SANG HO (KR)
PARK EUN KYUNG (KR)
LIM KWON JO (KR)
NAM SANG HYUN (KR)

International Classes:

C07D413/14; A61K31/538; A61P25/04

Foreign References:

US20050130962A1	2005-06-16
US6365736B1	2002-04-02
US4687770A	1987-08-18

Other References: