Title:
PHENETHYLNICOTINAMIDE COMPOUND
Document Type and Number:
WIPO Patent Application WO/2006/009054
Kind Code:
A1
Abstract:
[PROBLEMS] To provide a compound that is useful as a nitrogen monoxide production accelerator and/or endothelial nitrogen monoxide synthetic enzyme activator. [MEANS FOR SOLVING PROBLEMS] The phenethylnicotinamide compound as an active ingredient of proposed drugs exerts a bloodstream circulation improving effect according to excellent vascular endothelial nitrogen monoxide production accelerating potency and/or endothelial nitrogen monoxide synthetic enzyme activating potency. The proposed drugs are useful for relief of pathological conditions or diseases caused by vascular endothelial malfunction, especially as a therapeutic agent for peripheral arterial obstruction, arteriosclerosis, ischemic heart disease, etc.
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Inventors:
KAMIKUBO TAKASHI (JP)
MUKAI HANA (JP)
IBUKA RYOTARO (JP)
KOSHIO HIROYUKI (JP)
ISHIKAWA NORIKO (JP)
SHIBATA HIROSHI (JP)
SOGA YUMIKO (JP)
MUKAI HANA (JP)
IBUKA RYOTARO (JP)
KOSHIO HIROYUKI (JP)
ISHIKAWA NORIKO (JP)
SHIBATA HIROSHI (JP)
SOGA YUMIKO (JP)
Application Number:
PCT/JP2005/012991
Publication Date:
January 26, 2006
Filing Date:
July 14, 2005
Export Citation:
Assignee:
ASTELLAS PHARMA INC (JP)
KAMIKUBO TAKASHI (JP)
MUKAI HANA (JP)
IBUKA RYOTARO (JP)
KOSHIO HIROYUKI (JP)
ISHIKAWA NORIKO (JP)
SHIBATA HIROSHI (JP)
SOGA YUMIKO (JP)
KAMIKUBO TAKASHI (JP)
MUKAI HANA (JP)
IBUKA RYOTARO (JP)
KOSHIO HIROYUKI (JP)
ISHIKAWA NORIKO (JP)
SHIBATA HIROSHI (JP)
SOGA YUMIKO (JP)
International Classes:
A61K31/455; A61K31/50; A61K31/505; A61P9/00; A61P43/00; C07D213/82; C07D213/89; C07D237/24; C07D239/28; C07D401/12
Foreign References:
JP2004518719A | 2004-06-24 | |||
JP2004518722A | 2004-06-24 | |||
JP2004518720A | 2004-06-24 | |||
JP2004115507A | 2004-04-15 |
Attorney, Agent or Firm:
Morita, Hiroshi c/o Astellas Pharma Inc. (Intellectual Property 3, -11,
Nihonbashi-Honcho 2-chom, Chuo-ku Tokyo 11, JP)
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