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Patent Searching and Data


Title:
PREPARATION OF OSEMOZOTAN AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS, AND ITS INTERMEDIATE
Document Type and Number:
WIPO Patent Application WO/2010/000193
Kind Code:
A1
Abstract:
The invention provides a process for preparing osemozotan and its pharmaceutically acceptable salts. The invention also provides an intermediate, (2R)-N-[3-(1,3- benzodioxol-5-yloxy)propyl]-1,4-benzodioxin-2-formamide, used in the process and its preparation.

Inventors:
WANG YONG (CN)
ZHANG GUISEN (CN)
MA YANQIN (CN)
ZHOU YINGZHEN (CN)
ZHOU SHIXIA (CN)
PENG WEIJUAN (CN)
Application Number:
PCT/CN2009/072509
Publication Date:
January 07, 2010
Filing Date:
June 29, 2009
Export Citation:
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Assignee:
NHWA PHARMA CORP (CN)
WANG YONG (CN)
ZHANG GUISEN (CN)
MA YANQIN (CN)
ZHOU YINGZHEN (CN)
ZHOU SHIXIA (CN)
PENG WEIJUAN (CN)
International Classes:
C07D407/12; C07D319/20
Foreign References:
EP0446921B11998-09-30
JPS58219114A1983-12-20
EP0054304A11982-06-23
Attorney, Agent or Firm:
NTD PATENT & TRADEMARK AGENCY LIMITED BEIJING OFFICE (Block A Investment Plaza, 27 Jinrongdajie, Xicheng District, Beijing 0, CN)
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