Title:
PROCESS FOR THE PREPARATION OF COBICISTAT INTERMEDIATES
Document Type and Number:
WIPO Patent Application WO/2014/057498
Kind Code:
A3
Abstract:
The present invention relates to cobicistat intermediates, processes and further conversion to cobicistat with improved yield and quality.
Inventors:
RAMA SHANKAR
VADALI LAKSHMANA RAO
KONDA RAMESH BABU
JALDU RAVIKANTH
VEMAVARAPU GOVARDHANA PHANI SHARMA
PALLA VIJAY KUMAR
YERVA ESWARA REDDY
VADALI LAKSHMANA RAO
KONDA RAMESH BABU
JALDU RAVIKANTH
VEMAVARAPU GOVARDHANA PHANI SHARMA
PALLA VIJAY KUMAR
YERVA ESWARA REDDY
Application Number:
PCT/IN2013/000608
Publication Date:
June 19, 2014
Filing Date:
October 07, 2013
Export Citation:
Assignee:
MYLAN LAB LTD (IN)
RAMA SHANKAR
VADALI LAKSHMANA RAO
KONDA RAMESH BABU
JALDU RAVIKANTH
VEMAVARAPU GOVARDHANA PHANI SHARMA
PALLA VIJAY KUMAR
YERVA ESWARA REDDY
RAMA SHANKAR
VADALI LAKSHMANA RAO
KONDA RAMESH BABU
JALDU RAVIKANTH
VEMAVARAPU GOVARDHANA PHANI SHARMA
PALLA VIJAY KUMAR
YERVA ESWARA REDDY
International Classes:
C07D417/12; C07C307/06; C07D203/24
Domestic Patent References:
WO2010115000A2 | 2010-10-07 |
Other References:
JOANNE HANNAM ET AL: "Rapid and Selective Synthesis of Substituted 1,2,5-Thiadiazolidine 1,1-Dioxides", SYNLETT, vol. 2006, no. 6, 1 April 2006 (2006-04-01), pages 833 - 836, XP055097678, ISSN: 0936-5214, DOI: 10.1055/s-2006-939039
DATABASE REGISTRY [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; 30 September 2009 (2009-09-30), AURORA FINE CHEMICALS LLC, 7929-SILVERTON AVENUE, SUITE 609, SANDIEGO, CA, 92126, USA: "Aurora Building Blocks", XP002719126, Database accession no. 1178000-69-5
DATABASE REGISTRY [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; 30 September 2009 (2009-09-30), AURORA FINE CHEMICALS LLC, 7929-SILVERTON AVENUE, SUITE 609, SANDIEGO, CA, 92126, USA: "Aurora Building Blocks", XP002719126, Database accession no. 1178000-69-5
Attorney, Agent or Firm:
NARAHARI, Babu Ambati (Anrich Industrial EstateBollaram, Jinnaram Mandal, Medak Dist, Andhra Pradesh, IN)
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