Title:
PYRIMIDINYLBENZIMIDAZOLE AND TRIAZINYLBENZIMIDAZOLE DERIVATIVES AND AGRICULTURA/HORTICULTURAL BACTERICIDES
Document Type and Number:
WIPO Patent Application WO/2000/029404
Kind Code:
A1
Abstract:
Pyrimidinylbenzimidazole and triazinylbenzimidazole derivatives represented by general formula [I]; agricultural/horticultural bactericides containing the same as the active ingredient; and intermediates in producing the same represented by general formula [XV]. A represents N or CR?3¿; R?1¿ and R?2¿ independently represent each hydrogen, halogeno, C¿1-6? alkyl, C¿2-6? alkenyl, etc.; R?3¿ represents hydrogen, C¿1-6? alkyl, C¿1-6? alkoxy or halogeno; R?5¿ represents amino, nitro, etc.; X represents hydrogen, halogeno, nitro, cyano, etc.; Y represents halogeno, nitro, cyano, C¿1-6? alkyl, etc.; and n is 0 or an integer of 1 to 3.
More Like This:
Inventors:
SHIBATA MASARU (JP)
KAWAI KIYOSHI (JP)
MAKIHARA TAKECHI (JP)
YONEKURA NORIHISA (JP)
KAWASHIMA TAKAHIRO (JP)
SAKAI JUNETSU (JP)
MURAMATSU NORIMICHI (JP)
KAWAI KIYOSHI (JP)
MAKIHARA TAKECHI (JP)
YONEKURA NORIHISA (JP)
KAWASHIMA TAKAHIRO (JP)
SAKAI JUNETSU (JP)
MURAMATSU NORIMICHI (JP)
Application Number:
PCT/JP1999/006364
Publication Date:
May 25, 2000
Filing Date:
November 15, 1999
Export Citation:
Assignee:
KUMIAI CHEMICAL INDUSTRY CO (JP)
IHARA CHEMICAL IND CO (JP)
SHIBATA MASARU (JP)
KAWAI KIYOSHI (JP)
MAKIHARA TAKECHI (JP)
YONEKURA NORIHISA (JP)
KAWASHIMA TAKAHIRO (JP)
SAKAI JUNETSU (JP)
MURAMATSU NORIMICHI (JP)
IHARA CHEMICAL IND CO (JP)
SHIBATA MASARU (JP)
KAWAI KIYOSHI (JP)
MAKIHARA TAKECHI (JP)
YONEKURA NORIHISA (JP)
KAWASHIMA TAKAHIRO (JP)
SAKAI JUNETSU (JP)
MURAMATSU NORIMICHI (JP)
International Classes:
A01N43/54; A01N43/66; A01P3/00; C07D239/48; C07D251/42; C07D251/44; C07D251/46; C07D403/04; (IPC1-7): C07D403/04; C07D239/46; C07D251/42; C07D251/44; C07D251/46; A01N43/52; A01N43/66
Domestic Patent References:
| WO1999005138A1 | 1999-02-04 |
Foreign References:
| US5179098A | 1993-01-12 | |||
| US4698091A | 1987-10-06 | |||
| EP0945443A1 | 1999-09-29 | |||
| US5714509A | 1998-02-03 | |||
| US5739129A | 1998-04-14 | |||
| US4999046A | 1991-03-12 | |||
| US4973690A | 1990-11-27 | |||
| US4802909A | 1989-02-07 | |||
| US4659363A | 1987-04-21 | |||
| US4694009A | 1987-09-15 | |||
| DD151404A1 | 1981-10-21 | |||
| JPS5665804A | 1981-06-03 |
Other References:
FORLANI LUCIANO.: "Tautomerism of some amino aza-containing heterocycles", J. HETEROCYCL. CHEM.,, vol. 29, no. 6, October 1992 (1992-10-01) - November 1992 (1992-11-01), pages 1461 - 1464, XP002935562
OBARA YOSHIHIKO ET AL.: "Studies on the biological activity of heterocyclic compounds. Part IV. On the blinding activities and acute oral toxicities of aminobenzenes, pyrimidines, purines, amino-s-triazines and their related compounds in baby chicks", NIPPON NOGE KAGAKU KAISHI,, vol. 55, no. 12, 1981, pages 1205 - 1212, XP002935563
NAKAMURA KENJI ET AL.: "The N1-N2 migration of the s-triazinyl group of 4-substituted N1,N1-bis-(s-triazinyl)-o-phenyl-ene-diamines", BULL. CHEM. SOC. JAP.,, vol. 45, no. 10, 1972, pages 3140 - 3147, XP002935564
CHEMICAL ABSTRACTS, vol. 73, 1970, Columbus, Ohio, US; abstract no. 35337Z, page 327; XP002909883
See also references of EP 1132387A4
OBARA YOSHIHIKO ET AL.: "Studies on the biological activity of heterocyclic compounds. Part IV. On the blinding activities and acute oral toxicities of aminobenzenes, pyrimidines, purines, amino-s-triazines and their related compounds in baby chicks", NIPPON NOGE KAGAKU KAISHI,, vol. 55, no. 12, 1981, pages 1205 - 1212, XP002935563
NAKAMURA KENJI ET AL.: "The N1-N2 migration of the s-triazinyl group of 4-substituted N1,N1-bis-(s-triazinyl)-o-phenyl-ene-diamines", BULL. CHEM. SOC. JAP.,, vol. 45, no. 10, 1972, pages 3140 - 3147, XP002935564
CHEMICAL ABSTRACTS, vol. 73, 1970, Columbus, Ohio, US; abstract no. 35337Z, page 327; XP002909883
See also references of EP 1132387A4
Attorney, Agent or Firm:
Ogawa, Toshiharu (38 Kanda-Higashimatsushitach, Chiyoda-ku Tokyo, JP)
Download PDF: