Title:
RECEPTOR ANTAGONIST
Document Type and Number:
WIPO Patent Application WO/2004/091628
Kind Code:
A1
Abstract:
An agent for controlling the function of an RFRP receptor, characterized by containing either a compound represented by the formula (I) [wherein ring A represents an optionally substituted aromatic ring; ring B represents an optionally substituted benzene ring; X represents oxygen, S(O)n (n is an integer of 0 to 2), or NR3 (R3 represents hydrogen, an optionally substituted hydrocarbon group, or an optionally substituted heterocyclic group); and R1 and R2 each represents hydrogen, an optionally substituted hydrocarbon group, or an optionally substituted heterocyclic group] or a salt of the compound.
Inventors:
ITOH FUMIO (JP)
HINUMA SHUJI (JP)
KANZAKI NAOYUKI (JP)
MABUCHI HIROSHI (JP)
YOSHIDA HIROMI (JP)
MATSUMOTO HIROKAZU (JP)
WAKABAYASHI TAKESHI (JP)
HINUMA SHUJI (JP)
KANZAKI NAOYUKI (JP)
MABUCHI HIROSHI (JP)
YOSHIDA HIROMI (JP)
MATSUMOTO HIROKAZU (JP)
WAKABAYASHI TAKESHI (JP)
Application Number:
PCT/JP2004/005406
Publication Date:
October 28, 2004
Filing Date:
April 15, 2004
Export Citation:
Assignee:
TAKEDA PHARMACEUTICAL (JP)
ITOH FUMIO (JP)
HINUMA SHUJI (JP)
KANZAKI NAOYUKI (JP)
MABUCHI HIROSHI (JP)
YOSHIDA HIROMI (JP)
MATSUMOTO HIROKAZU (JP)
WAKABAYASHI TAKESHI (JP)
ITOH FUMIO (JP)
HINUMA SHUJI (JP)
KANZAKI NAOYUKI (JP)
MABUCHI HIROSHI (JP)
YOSHIDA HIROMI (JP)
MATSUMOTO HIROKAZU (JP)
WAKABAYASHI TAKESHI (JP)
International Classes:
A61P1/14; A61P3/06; A61P3/10; A61P5/24; A61P7/00; A61P7/02; A61P9/10; A61P13/02; A61P15/00; A61P17/00; A61P19/02; A61P19/08; A61P21/00; A61P25/04; A61P25/08; A61P25/14; A61P25/28; A61P35/00; A61P37/06; A61P43/00; C07D267/08; (IPC1-7): A61K31/5513; A61K31/553; A61K31/5377; A61P43/00; A61P25/04; A61P37/06; A61P35/00; A61P15/00; A61P9/10; A61P7/02; A61P1/14; A61P25/28; A61P21/00; A61P25/08; A61P25/14; A61P7/00; A61P5/24; A61P3/10; A61P13/02; A61P3/06; A61P17/00; A61P19/02; A61P19/08; C07D267/14; C07D243/24; C07D281/08; C07D413/12
Domestic Patent References:
WO1998047882A1 | 1998-10-29 | |||
WO1997010224A1 | 1997-03-20 | |||
WO2001055121A1 | 2001-08-02 | |||
WO2003018795A1 | 2003-03-06 |
Foreign References:
JP2002080468A | 2002-03-19 | |||
JP2003081873A | 2003-03-19 |
Attorney, Agent or Firm:
Takahashi, Shuichi c/o Osaka Plant of TAKEDA CHEMICAL INDUSTRIES LTD. (17-85, Jusohonmachi 2-chome, Yodogawa-ku, Osaka-sh, Osaka 24, JP)
Download PDF: