Title:
SIX-MEMBERED AROMATIC RING-PYRROLIDONE DERIVATIVE, AND PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2023/165551
Kind Code:
A1
Abstract:
The present application relates to a six-membered aromatic ring-pyrrolidone derivative, and a pharmaceutical composition thereof and the use thereof. The six-membered aromatic ring-pyrrolidone derivative has the structure as shown in formula (I).
Inventors:
SUN HONGPENG (CN)
XU FENG (CN)
WANG HAILONG (CN)
XI BAOXIN (CN)
TONG ZHONGAN (CN)
MA QIAN (CN)
XU FENG (CN)
WANG HAILONG (CN)
XI BAOXIN (CN)
TONG ZHONGAN (CN)
MA QIAN (CN)
Application Number:
PCT/CN2023/079240
Publication Date:
September 07, 2023
Filing Date:
March 02, 2023
Export Citation:
Assignee:
SHANGHAI HAIYAN PHARMACEUTICAL TECH CO LTD (CN)
YANGTZE RIVER PHARM GROUP CO (CN)
YANGTZE RIVER PHARM GROUP CO (CN)
International Classes:
A61K31/427; C07D417/04; A61K31/4985; A61P3/00; A61P29/00; A61P35/00; C07D487/04
Domestic Patent References:
WO2022017371A1 | 2022-01-27 | |||
WO2020247496A1 | 2020-12-10 | |||
WO2020102216A1 | 2020-05-22 |
Foreign References:
CN114025756A | 2022-02-08 |
Other References:
MILES DILLON H., YAN XUELEI, THOMAS-TRAN RHIANNON, FOURNIER JEREMY, SHARIF EHESAN U., DREW SAMUEL L., MATA GUILLAUME, LAWSON KENNE: "Discovery of Potent and Selective 7-Azaindole Isoindolinone-Based PI3Kγ Inhibitors", ACS MEDICINAL CHEMISTRY LETTERS, AMERICAN CHEMICAL SOCIETY, US, vol. 11, no. 11, 12 November 2020 (2020-11-12), US , pages 2244 - 2252, XP055954608, ISSN: 1948-5875, DOI: 10.1021/acsmedchemlett.0c00387
Attorney, Agent or Firm:
ADVANCE CHINA IP LAW OFFICE (CN)
Download PDF: