Title:
THIADIAZOLE DERIVATIVES, PESTICIDES FOR AGRICULTURAL AND HORTICULTURAL USE AND USAGE THEREOF
Document Type and Number:
WIPO Patent Application WO/2002/092584
Kind Code:
A1
Abstract:
Thiadiazole derivatives represented by the general formula (I); pesticides for agricultural and horticultural use, containing the compounds as the active ingredient; and usage thereof: (II) wherein R is hydrogen, cyano, nitro, C¿1-6? alkyl, C¿3-6? cycloalkyl, substituted C¿1-6? alkyl, or the like; Y is halogeno, C¿1-6? alkyl, C¿1-6? haloalkyl, or the like; Z is oxygen or sulfur; A is a group represented by the general formula (II); W is carbon or nitrogen; and Q is T-U (wherein T is -O-, -S-, -CH¿2?-, or the like; and U is hydrogen, C¿1-6? alkyl, or the like).
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Inventors:
NAKAO HAYAMI (JP)
MATSUZAKI YOSHIHIRO (JP)
TOHNISHI MASANORI (JP)
MORIMOTO MASAYUKI (JP)
FUJIOKA SHINSUKE (JP)
TAKEMOTO TSUYOSHI (JP)
MAMEZUKA KOKI (JP)
MATSUZAKI YOSHIHIRO (JP)
TOHNISHI MASANORI (JP)
MORIMOTO MASAYUKI (JP)
FUJIOKA SHINSUKE (JP)
TAKEMOTO TSUYOSHI (JP)
MAMEZUKA KOKI (JP)
Application Number:
PCT/JP2002/004592
Publication Date:
November 21, 2002
Filing Date:
May 13, 2002
Export Citation:
Assignee:
NIHON NOHYAKU CO LTD (JP)
NAKAO HAYAMI (JP)
MATSUZAKI YOSHIHIRO (JP)
TOHNISHI MASANORI (JP)
MORIMOTO MASAYUKI (JP)
FUJIOKA SHINSUKE (JP)
TAKEMOTO TSUYOSHI (JP)
MAMEZUKA KOKI (JP)
NAKAO HAYAMI (JP)
MATSUZAKI YOSHIHIRO (JP)
TOHNISHI MASANORI (JP)
MORIMOTO MASAYUKI (JP)
FUJIOKA SHINSUKE (JP)
TAKEMOTO TSUYOSHI (JP)
MAMEZUKA KOKI (JP)
International Classes:
A01N43/82; A01N43/824; A01N47/20; A01N47/32; C07D285/135; C07D417/12; C07D285/12; (IPC1-7): C07D285/135; A01N43/824; C07D417/12
Foreign References:
| JPS4823935A | ||||
| US4416683A | 1983-11-22 | |||
| JPH01113369A | 1989-05-02 | |||
| US4141984A | 1979-02-27 | |||
| JPS60223067A | 1985-11-07 | |||
| JPS56158703A | 1981-12-07 | |||
| JP2000226389A | 2000-08-15 |
Other References:
YOSHIAKI NAKAGAWA ET AL.: "Quantitative structure-activity relationships of larvicidal N-(5-(substituted phenyl)-1,3,4-thiadiazol-2-yl)-benzamides in the inhibition of N-acetyl glucosamine incorporation into a cultured integument system", J. PESTICIDE SCI., vol. 21, no. 2, 1996, pages 195 - 201, XP002956628
FENG C.C. ET AL.: "Multidrug analysis of some insect growth regulators by reserved-phase high-performance liquid chromatography", J. LIQUID CHROMATOGR., vol. 7, no. 1, 1984, pages 95 - 109, XP002956629
WHITE G.A. ET AL.: "Substituted 2-methylbenzanilides and structurally related carboxamides: inhibition of complex II activity in mitochondria from a wild-type strain and a carboxin-resistant mutation strain of ustilago maydis", OESTIVIDE BIOCHEMISTRY AND PHYSIOLOGY, vol. 34, no. 3, 1989, pages 255 - 276, XP002956630
DAIDONE G. ET AL.: "Salicylanilide and its heterocyclic analogues. A comparative study of their antimicrobial activity", PHARMAZIE, vol. 45, no. 6, 1990, pages 441 - 442, XP002956631
LUKES JAMES J. ET AL.: "Substituted thiadiazolines as inhibitors of central nervous system carbonic anhydrase", J. MED. CHEM., vol. 18, no. 4, 1975, pages 351 - 354, XP002956632
COBURN ROBERT A. ET AL.: "Potential salicylamide antiplaque agents: in vitro antibacterial activity against actinomyces viscosus", J. MED. CHEM., vol. 24, no. 10, 1981, pages 1245 - 1249, XP000992845
DATABASE CAPLUS [online] WANG Y. ET AL.: "Synthesis of 5-(3-pyridyl)-2-aroylamino-1,3,4-thiadiazole derivatives", XP002957314, Database accession no. 2001:461281
DATABASE CAPLUS [online] SHAMS-EL-DINE SH.A. ET AL.: "Chemical studies in the field of oral hypoglycemic agents. III.", XP002957315, Database accession no. 1975:531514
FENG C.C. ET AL.: "Multidrug analysis of some insect growth regulators by reserved-phase high-performance liquid chromatography", J. LIQUID CHROMATOGR., vol. 7, no. 1, 1984, pages 95 - 109, XP002956629
WHITE G.A. ET AL.: "Substituted 2-methylbenzanilides and structurally related carboxamides: inhibition of complex II activity in mitochondria from a wild-type strain and a carboxin-resistant mutation strain of ustilago maydis", OESTIVIDE BIOCHEMISTRY AND PHYSIOLOGY, vol. 34, no. 3, 1989, pages 255 - 276, XP002956630
DAIDONE G. ET AL.: "Salicylanilide and its heterocyclic analogues. A comparative study of their antimicrobial activity", PHARMAZIE, vol. 45, no. 6, 1990, pages 441 - 442, XP002956631
LUKES JAMES J. ET AL.: "Substituted thiadiazolines as inhibitors of central nervous system carbonic anhydrase", J. MED. CHEM., vol. 18, no. 4, 1975, pages 351 - 354, XP002956632
COBURN ROBERT A. ET AL.: "Potential salicylamide antiplaque agents: in vitro antibacterial activity against actinomyces viscosus", J. MED. CHEM., vol. 24, no. 10, 1981, pages 1245 - 1249, XP000992845
DATABASE CAPLUS [online] WANG Y. ET AL.: "Synthesis of 5-(3-pyridyl)-2-aroylamino-1,3,4-thiadiazole derivatives", XP002957314, Database accession no. 2001:461281
DATABASE CAPLUS [online] SHAMS-EL-DINE SH.A. ET AL.: "Chemical studies in the field of oral hypoglycemic agents. III.", XP002957315, Database accession no. 1975:531514
Attorney, Agent or Firm:
Asamura, Kiyoshi (New Ohtemachi Bldg. 2-1, Ohtemachi 2-chom, Chiyoda-ku Tokyo, JP)
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