Title:
THIOALKYLAMINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF
Document Type and Number:
WIPO Patent Application WO/2001/023350
Kind Code:
A1
Abstract:
Thioalkylamine derivatives represented by general formula (I); and a process for the preparation thereof wherein R¿1? and R¿2? are each H, (C¿1-4?)alkyl, (C¿3-8?)cycloalkyl, (C¿3-8?)cycloalkyl(C¿1-4?)alkyl, (substituted) phenyl, (substituted) phenyl(C¿1-4?)alkyl, or the like; R¿3? and R¿4? are each H or (C¿1-4?)alkyl; R¿5? and R¿6? are each H, (C¿1-4?)alkyl, (substituted) phenyl, or (substituted) phenyl(C¿1-4?)alkyl; alternatively R¿1? and R¿2?, R¿1? and R¿3? or R¿5?, R¿3? and R¿4?, R¿3? and R¿5?, or R¿5? and R¿6? may together form lower alkylene; and R is (C¿1-12?)alkyl, (C¿3-8?)cycloalkyl, (C¿3-8?)cycloalkyl(C¿1-4?)alkyl, (substituted) phenyl, (substituted) phenyl(C¿1-4?)alkyl, naphthyl, a (substituted) aromatic heterocycle, or the like.
More Like This:
Inventors:
SANPEI OSAMU (JP)
TSUBATA KENJI (JP)
TSUBATA KENJI (JP)
Application Number:
PCT/JP2000/006673
Publication Date:
April 05, 2001
Filing Date:
September 27, 2000
Export Citation:
Assignee:
NIHON NOHYAKU CO LTD (JP)
SANPEI OSAMU (JP)
TSUBATA KENJI (JP)
SANPEI OSAMU (JP)
TSUBATA KENJI (JP)
International Classes:
C07C319/14; C07C323/25; C07D213/70; C07D213/89; C07D249/12; C07D295/088; C07D333/34; (IPC1-7): C07C323/25; C07D213/70; C07D295/08; C07D333/34; C07D213/89; C07C319/14
Domestic Patent References:
WO1999050238A1 | 1999-10-07 | |||
WO1995000493A1 | 1995-01-05 | |||
WO1989010919A1 | 1989-11-16 |
Foreign References:
EP0468434A1 | 1992-01-29 | |||
EP0066993A1 | 1982-12-15 | |||
EP0066415A2 | 1982-12-08 | |||
EP0053015A1 | 1982-06-02 | |||
US4259334A | 1981-03-31 | |||
GB1604674A | 1981-12-16 | |||
GB1469772A | 1977-04-06 | |||
GB1527510A | 1978-10-04 | |||
US5405947A | 1995-04-11 |
Other References:
See also references of EP 1216988A4
Attorney, Agent or Firm:
Asamura, Kiyoshi (Room 331 2-1, Ohtemachi 2-chom, Chiyoda-ku Tokyo, JP)
Download PDF: