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Title:
TREATING RESPIRATORY DISEASES WITH GYCOPYRROLATE AND ANALOGUES
Document Type and Number:
WIPO Patent Application WO/2005/107872
Kind Code:
A2
Abstract:
Glycopyrrate or an analogue thereof is useful for the treatment of bronchospasm or as a rescue medication.

Inventors:
SNAPE SUSAN (GB)
BANNISTER ROBIN MARK (GB)
Application Number:
PCT/GB2005/001776
Publication Date:
November 17, 2005
Filing Date:
May 10, 2005
Export Citation:
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Assignee:
ARAKIS LTD (GB)
SNAPE SUSAN (GB)
BANNISTER ROBIN MARK (GB)
International Classes:
A61K31/00; A61K31/352; A61K31/40; A61K31/465; (IPC1-7): A61P11/00; A61P11/08; A61K31/40
Domestic Patent References:
WO2001076575A22001-10-18
WO2005074900A22005-08-18
Other References:
WALKER F B ET AL: "PROLONGED EFFECT OF INHALED GLYCOPYRROLATE IN ASTHMA" CHEST, THE COLLEGE, CHICAGO, IL, US, vol. 91, no. 1, January 1987 (1987-01), pages 49-51, XP000979963 ISSN: 0012-3692 cited in the application
SKORODIN M S: "PHARMACOTHERAPY FOR ASTHMA AND CHRONIC OBSTRUCTIVE PULMONARY DISEASE CURRENT THINKING, PRACTICES, AND CONTROVERSIES" ARCHIVES OF INTERNAL MEDICINE, AMERICAN MEDICAL ASSOCIATION, CHICAGO, IL, US, vol. 153, no. 7, 12 April 1993 (1993-04-12), pages 814-828, XP000979854 ISSN: 0003-9926 cited in the application
SELF T ET AL: "Glycopyrrolate for asthma." THE AMERICAN JOURNAL OF EMERGENCY MEDICINE. JUL 1992, vol. 10, no. 4, July 1992 (1992-07), pages 395-396, XP008057576 ISSN: 0735-6757
CYDULKA ET AL: "Effects of Combined Treatment With Glycopyrrolate and Albuterol in Acute Exacerbation of Chronic Obstructive Pulmonary Disease" ANNALS OF EMERGENCY MEDICINE, LANSING, MI, US, vol. 25, no. 4, April 1995 (1995-04), pages 470-473, XP005127538 ISSN: 0196-0644
BROCK-UTNE J G: "Reversal of neuromuscular blockade by glycopyrrolate and neostigmine. A study of the effects on lower oesophageal sphincter tone." ANAESTHESIA. 1979 JUL-AUG, vol. 34, no. 7, July 1979 (1979-07), pages 620-623, XP008057585 ISSN: 0003-2409
MAESEN F P V ET AL: "TIOTROPIUM BROMIDE, A NEW LONG-ACTING ANTIMUSCARINIC BRONCHODILATOR: A PHARMACODYNAMIC STUDY IN PATIENTS WITH CHRONIC OBSTRUCTIVE PULMONARY DISEASE (COPD)" EUROPEAN RESPIRATORY JOURNAL, MUNKSGAARD INTERNATIONAL PUBLISHERS, COPENHAGEN, DK, vol. 8, no. 9, September 1995 (1995-09), pages 1506-1513, XP001118564 ISSN: 0903-1936 cited in the application
Attorney, Agent or Firm:
GILL JENNINGS & EVERY LLP (7 Eldon Street, London EC2M 7LH, GB)
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