TRYASOLYL TROPANE DERIVATIVES AS CCR5 MODULATORS

WIPO Patent Application WO2001090106

A3

The present invention provides compounds of the formula (I): wherein R<1> is C3-6 cycloalkyl optionally substituted by one or more fluorine atoms, or C1-6 alkyl optionally substituted by one or more fluorine atoms, or C3-6 cycloalkylmethyl optionally ring-substituted by one or more fluorine atoms; and R<2> is phenyl optionally substituted by one or more fluorine atoms, to pharmaceutically acceptable salts and solvates thereof, and to processes for the preparation of, intermediates used in the preparation of, compositions containing and the uses of, such compounds.

PERROS MANOUSSOS (GB)
PRICE DAVID ANTHONY (GB)
STAMMEN BLANDA LUZIA CHRISTA (GB)
WOOD ANTHONY (GB)

PCT/IB2001/000806

March 28, 2002

May 09, 2001

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PFIZER LTD (GB)
PFIZER (US)
PERROS MANOUSSOS (GB)
PRICE DAVID ANTHONY (GB)
STAMMEN BLANDA LUZIA CHRISTA (GB)
WOOD ANTHONY (GB)

A61K31/4196; A61K31/46; A61P1/04; A61P1/12; A61P1/18; A61P3/10; A61P9/04; A61P11/00; A61P11/06; A61P11/08; A61P13/12; A61P15/00; A61P25/00; A61P25/28; A61P27/16; A61P29/00; A61P31/18; A61P37/00; A61P37/06; A61P43/00; C07B53/00; C07B61/00; C07C233/60; C07C233/61; C07C233/63; C07D451/04; C07D; (IPC1-7): C07D451/04; A61K31/46; A61P29/00; A61P31/18

WO1998025617A1	1998-06-18
WO2000038680A1	2000-07-06
WO1999004794A1	1999-02-04
WO1997019060A1	1997-05-29
WO1998025604A1	1998-06-18
WO1999017773A1	1999-04-15
WO1998002151A2	1998-01-22
WO1999037617A1	1999-07-29
WO1999037619A1	1999-07-29
WO1997024325A1	1997-07-10

EP0903349A2	1999-03-24
EP0630887A1	1994-12-28

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