UREA ANTAGONISTS OF P2Y1 RECEPTOR USEFUL IN THE TREATMENT OF THROMBOTIC CONDITIONS

WIPO Patent Application WO2005113511

A9

The present invention provides novel pyridyl or phenyl ureas and analogues thereof, which are selective inhibitors of the human P2Y₁ receptor. The invention also provides for various pharmaceutical compositions of the same and methods for treating diseases responsive to modulation of P2Y₁ receptor activity.

CHAO HANNGUANG J (US)
TUERDI HUJI (US)
HERPIN TIMOTHY (US)
ROBERGE JACQUES YVES (US)
LIU YALEI (US)
LAWRENCE R MICHAEL (US)
REHFUSS ROBERT P (US)
CLARK CHARLES G (US)
QIAO JENNIFER X (US)
GUNGOR TIMUR (US)
LAM PATRICK Y S (US)
WANG TAMMY C (US)
RUEL REJEAN (CA)
L HEUREUX ALEXANDRE L (CA)
THIBEAULT CARL (CA)
BOUTHILLIER GILLES (CA)
SCHNUR DORA M (US)

PCT/US2005/016422

February 02, 2006

May 11, 2005

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BRISTOL MYERS SQUIBB CO (US)
CHAO HANNGUANG J (US)
TUERDI HUJI (US)
HERPIN TIMOTHY (US)
ROBERGE JACQUES YVES (US)
LIU YALEI (US)
LAWRENCE R MICHAEL (US)
REHFUSS ROBERT P (US)
CLARK CHARLES G (US)
QIAO JENNIFER X (US)
GUNGOR TIMUR (US)
LAM PATRICK Y S (US)
WANG TAMMY C (US)
RUEL REJEAN (CA)
L HEUREUX ALEXANDRE L (CA)
THIBEAULT CARL (CA)
BOUTHILLIER GILLES (CA)
SCHNUR DORA M (US)

A61K31/4439; A61K31/444; A61K31/501; C07C275/30; C07C275/32; C07D213/40; C07D213/75; C07D213/89; C07D231/40; C07D231/50; C07D237/22; C07D333/36; C07D401/12; C07D401/14; C07D405/12; C07D405/14; C07D409/12; C07D409/14; C07D413/12; C07D417/12; C07F7/18; (IPC1-7): C07D231/50; C07D231/40; C07D213/40; C07D413/12; C07D401/12; C07D405/12; C07D417/12; C07D333/36; A61K31/444; A61P7/02

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