Title:
シクロヘキシルアミン類
Document Type and Number:
Japanese Patent JP6495654
Kind Code:
B2
Abstract:
The present application provides novel compounds and methods for preparing and using these compounds. These compounds are useful in treating pain, itch, overactive bladder and/or interstitial cystitis in patients by administering one or more of the compounds to a patient. The methods include administering a compound of formula (I) and a TRPV1 receptor activator. In one embodiment, the TRPV1 receptor activator is lidocaine.
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Inventors:
Scott Kevin Thompson
Roger Astbury Smith
Sandeep Gupta
Tony Priestley
Nicholas James Laping
Assis K. Saha
Sonali Rudra
Roger Astbury Smith
Sandeep Gupta
Tony Priestley
Nicholas James Laping
Assis K. Saha
Sonali Rudra
Application Number:
JP2014538934A
Publication Date:
April 03, 2019
Filing Date:
October 24, 2012
Export Citation:
Assignee:
Asana Biosciences, Limited Liability Company
International Classes:
A61K31/167; C07C219/14; A61K31/235; A61K31/351; A61K31/381; A61K31/40; A61K31/4025; A61K31/452; A61K31/4535; A61K45/00; A61P13/10; A61P17/04; A61P25/04; A61P43/00; C07D207/34; C07D295/088; C07D309/14; C07D333/38; C07D333/70
Domestic Patent References:
JP472623B1 |
Other References:
Acta Pharm.Suec.,(1984),Vol.21,No.5,pp.271-294
Cellular and Molecular Basis of Cholinergic Function (1987),pp.347-354
IZVESTIYA AKADEMII NAUK ARMYANSKOI SSR,KHIMICHESKIE NAUKI,(1963),16(2),pp.163-174
Cellular and Molecular Basis of Cholinergic Function (1987),pp.347-354
IZVESTIYA AKADEMII NAUK ARMYANSKOI SSR,KHIMICHESKIE NAUKI,(1963),16(2),pp.163-174
Attorney, Agent or Firm:
Atsushi Aoki
Takashi Ishida
Fukumoto product
Tetsuji Koga
Yoichi Watanabe
Masaru Nakajima
Ryotaro Takei
Takashi Ishida
Fukumoto product
Tetsuji Koga
Yoichi Watanabe
Masaru Nakajima
Ryotaro Takei